SCHEMBL6973461

SCHEMBL6973461

CC(=O)OCc1nc(C(C)C)c(Sc2cc(F)cc(F)c2)n1Cc1ccccn1

nearest known ligand 0.39

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 14/20 0.39
SYK P43405 1/20 0.35
GRM5 P41594 1/20 0.34
ENPP2 Q13822 1/20 0.34
MEN1 O00255 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GFER P55789 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7084823 0.93 S1PR3 (0.39) S1PR3SYKGRM5ENPP2MEN1
SCHEMBL6968357 0.92 S1PR3 (0.37) S1PR3SYKKDM4EALDH1A1LMNA
SCHEMBL7084640 0.92 S1PR3 (0.39) S1PR3SYKGRM5ENPP2KDM4E
SCHEMBL7084180 0.91 S1PR3 (0.39) S1PR3ENPP2LMNA
SCHEMBL7084491 0.90 CYP1A2 (0.40) SYKMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL7078972 0.89 SLC16A3 (0.35) S1PR3GRM5MEN1CYP1A2CYP2C9
SCHEMBL7082232 0.87 S1PR3 (0.36) S1PR3ENPP2
SCHEMBL6961563 0.87 S1PR3 (0.37) S1PR3GRM5
SCHEMBL6973222 0.86 S1PR3 (0.41) S1PR3ALDH1A1
SCHEMBL7081153 0.86 MAPT (0.39) GRM5MEN1CYP1A2CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed