SCHEMBL7084640

SCHEMBL7084640

CC(C)c1nc(COC(N)=O)n(Cc2ccccn2)c1Sc1cc(F)cc(F)c1

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 12/20 0.39
GRM5 P41594 1/20 0.34
PLA2G2A P14555 1/20 0.34
ENPP2 Q13822 1/20 0.34
TLR7 Q9NYK1 1/20 0.33
SYK P43405 1/20 0.33
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
LMNA P02545 1/20 0.33
GFER P55789 1/20 0.33
OPRM1 P35372 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7078713 0.93 S1PR3 (0.39) S1PR3GRM5PLA2G2AENPP2
SCHEMBL6961563 0.93 S1PR3 (0.37) S1PR3GRM5PLA2G2ATLR7
SCHEMBL6973461 0.92 S1PR3 (0.39) S1PR3GRM5ENPP2SYKKDM4E
SCHEMBL6972492 0.91 S1PR3 (0.38) S1PR3PLA2G2AKDM4EALDH1A1LMNA
SCHEMBL7082317 0.90 PLA2G2A (0.36) S1PR3PLA2G2ATLR7KDM4EALDH1A1
SCHEMBL6967024 0.90 ALDH1A1 (0.35) PLA2G2ATLR7KDM4EALDH1A1LMNA
SCHEMBL6972895 0.90 S1PR3 (0.37) S1PR3PLA2G2ATLR7KDM4EALDH1A1
SCHEMBL7084180 0.90 S1PR3 (0.39) S1PR3ENPP2LMNA
SCHEMBL6966022 0.90 ADRA1D (0.36) S1PR3GRM5PLA2G2ATLR7KDM4E
SCHEMBL6975183 0.87 ENPP2 (0.35) PLA2G2AENPP2TLR7KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed