SCHEMBL6973575

SCHEMBL6973575

Nc1cc(N)c(Cl)c(S(=O)(=O)c2cccc3cnccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 6/20 0.47
CYP2D6 P10635 5/20 0.47
LMNA P02545 3/20 0.47
CYP1A2 P05177 2/20 0.47
CYP2C19 P33261 2/20 0.47
CYP2C9 P11712 1/20 0.47
PRKD3 O94806 5/20 0.46
PRKCG P05129 5/20 0.46
PRKCB P05771 5/20 0.46
PRKCA P17252 5/20 0.46
PRKCH P24723 5/20 0.46
PRKCI P41743 5/20 0.46
PRKCE Q02156 5/20 0.46
PRKCQ Q04759 5/20 0.46
PRKCZ Q05513 5/20 0.46
PRKCD Q05655 5/20 0.46
PRKD1 Q15139 5/20 0.46
PRKACA P17612 4/20 0.46
PRKACG P22612 4/20 0.46
PRKACB P22694 4/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6971281 0.85 CYP3A4 (0.47) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6973402 0.84 CYP3A4 (0.51) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6974826 0.82 CYP3A4 (0.48) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6968810 0.82 CYP3A4 (0.49) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6967362 0.81 CYP3A4 (0.59) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6974061 0.77 CYP3A4 (0.44) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6959712 0.77 CYP3A4 (0.49) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6963108 0.76 HTR6 (0.68) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6967123 0.75 CYP3A4 (0.50) CYP3A4CYP2D6LMNACYP1A2CYP2C19
SCHEMBL6962005 0.75 NPY1R (0.43) CYP3A4CYP2D6LMNACYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0855391-B1 NOVEL ISOQUINOLINE DERIVATIVES DAIICHI SEIYAKU CO (JP) 2003-10-15 EP disclosed
US-5959107-A Isoquinoline derivatives SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1999-09-28 US disclosed
EP-0855391-A1 NOVEL ISOQUINOLINE DERIVATIVES SNOW BRAND MILK PRODUCTS CO., LTD. (JP) 1998-07-29 EP disclosed