SCHEMBL6975571

SCHEMBL6975571

OCCc1coc(-c2ccc(Br)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.49
HDAC8 Q9BY41 2/20 0.49
HDAC6 Q9UBN7 2/20 0.49
PDE4B Q07343 2/20 0.41
LMNA P02545 1/20 0.38
TSHR P16473 2/20 0.37
KDM4E B2RXH2 1/20 0.37
NPC1 O15118 1/20 0.37
MAPT P10636 1/20 0.37
RAB9A P51151 1/20 0.37
HSD17B10 Q99714 1/20 0.37
NR1H4 Q96RI1 1/20 0.37
SMPD1 P17405 1/20 0.36
DRD2 P14416 1/20 0.36
DRD4 P21917 1/20 0.36
DRD3 P35462 1/20 0.36
GAA P10253 1/20 0.36
KMT2A Q03164 1/20 0.36
FFAR1 O14842 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2225047 0.83 HDAC1 (0.45) HDAC1HDAC8HDAC6PDE4BLMNA
SCHEMBL27682910 0.83 DRD2 (0.49) HDAC1HDAC8HDAC6LMNATSHR
SCHEMBL5229185 0.83 HDAC1 (0.48) HDAC1HDAC8HDAC6PDE4B
SCHEMBL5106193 0.83 DRD2 (0.51) HDAC1HDAC8HDAC6LMNATSHR
SCHEMBL4906065 0.80 IKBKB (0.41) LMNATSHRKDM4ENPC1MAPT
SCHEMBL4905721 0.80 PPARG (0.49) LMNATSHRKDM4EHSD17B10GAA
SCHEMBL2225496 0.79 HDAC1 (0.47) HDAC1HDAC8HDAC6PDE4BLMNA
SCHEMBL6971893 0.78 HDAC1 (0.54) HDAC1HDAC8HDAC6PDE4BLMNA
SCHEMBL5119297 0.76 HDAC1 (0.51) HDAC1HDAC8HDAC6LMNATSHR
SCHEMBL31163804 0.76 CYP1A2 (0.37) LMNATSHRNPC1MAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1206457-B1 BIARYL-OXA(THIA)ZOLE DERIVATIVES AND THEIR USE AS PPARS MODULATORS LILLY CO ELI (US) 2003-10-15 EP claimed