SCHEMBL6976955

SCHEMBL6976955

CC(C)c1nc(C(O)Cc2ccccn2)[nH]c1Sc1cc(Cl)cc(Cl)c1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 1/20 0.34
PTPRA P18433 1/20 0.33
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
ALDH1A1 P00352 3/20 0.32
KDM4E B2RXH2 2/20 0.32
MAPT P10636 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
CCNE2 O96020 1/20 0.31
CDK4 P11802 1/20 0.31
CCND1 P24385 1/20 0.31
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
FDPS P14324 1/20 0.31
XIAP P98170 1/20 0.31
BIRC2 Q13490 1/20 0.31
MC4R P32245 1/20 0.31
CYP1A2 P05177 1/20 0.30
CYP2C19 P33261 1/20 0.30
GRM4 Q14833 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7079932 0.92 GRM5 (0.38) PTPRAMEN1KMT2AALDH1A1KDM4E
SCHEMBL7081552 0.89 PTPRA (0.34) PTPRAKMT2AALDH1A1KDM4EFDPS
SCHEMBL6963979 0.88 PTPRA (0.39) PTPRAKMT2AALDH1A1KDM4EMAPT
SCHEMBL6973516 0.88 PTPRA (0.33) PTPRAALDH1A1KDM4EFDPSCYP1A2
SCHEMBL6966853 0.86 TDP1 (0.33) RHEBKMT2A
SCHEMBL6967986 0.84 SLC6A9 (0.34) PTPRAKMT2AALDH1A1KDM4EMAPT
SCHEMBL6966456 0.84
SCHEMBL7078977 0.84 RHEB (0.34) RHEBPTPRAMEN1KMT2AALDH1A1
SCHEMBL7164320 0.84 RHEB (0.31) RHEB
SCHEMBL6973238 0.83 CYP1A2 (0.33) CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed