SCHEMBL6963979

SCHEMBL6963979

CC(C)c1nc(C(O)Cc2ccccn2)[nH]c1Sc1ccccc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRA P18433 1/20 0.39
KDM4E B2RXH2 1/20 0.36
GRIN2D O15399 1/20 0.35
GRIN3B O60391 1/20 0.35
GRIN1 Q05586 1/20 0.35
GRIN2A Q12879 1/20 0.35
GRIN2B Q13224 1/20 0.35
GRIN2C Q14957 1/20 0.35
GRIN3A Q8TCU5 1/20 0.35
DHFR P00374 1/20 0.34
FDPS P14324 1/20 0.34
CYP1A2 P05177 5/20 0.33
CYP2D6 P10635 3/20 0.33
TSHR P16473 2/20 0.33
MAPT P10636 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 3/20 0.33
CYP2C19 P33261 2/20 0.33
SLC6A4 P31645 1/20 0.32
FNTA P49354 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7081552 0.89 PTPRA (0.34) PTPRAKDM4EFDPSCYP1A2CYP2D6
SCHEMBL6967986 0.89 SLC6A9 (0.34) PTPRAKDM4EGRIN1GRIN2BFDPS
SCHEMBL7079932 0.89 GRM5 (0.38) PTPRAKDM4ECYP1A2MAPTSMN1; SMN2
SCHEMBL6973516 0.88 PTPRA (0.33) PTPRAKDM4EFDPSCYP1A2ALDH1A1
SCHEMBL6976955 0.88 RHEB (0.34) PTPRAKDM4EFDPSCYP1A2MAPT
SCHEMBL6972933 0.85 CYP1A2 (0.39) KDM4ECYP1A2MAPTSMN1; SMN2ALDH1A1
SCHEMBL7078351 0.84 SLC6A4 (0.36) DHFRCYP1A2CYP2D6ALDH1A1CYP2C19
SCHEMBL7084495 0.82 PTPRA (0.37) PTPRADHFRFDPSCYP1A2CYP2D6
SCHEMBL6974559 0.82 PTPRA (0.32) PTPRAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL7081802 0.82 DHFR (0.39) KDM4EDHFRSLC6A4KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0786455-B1 IMIDAZOLE DERIVATIVE SHIONOGI & CO (JP) 2003-12-03 EP disclosed
US-6147097-A METHOD FOR TREATING AIDS SHIONOGI & CO., LTD. (JP) 2000-11-14 US disclosed
US-5910506-A IMIDAZOLE DERIVATIVES, E.G.5-(3,5-DICHLOROPHENYLTHIO)-1,2-DIMETHYL-4-ISOPROPYL-1H-IMIDAZOLE; VIRICIDES; AIDS; NONTOXIC SHIONOGI & CO., LTD. (JP) 1999-06-08 US disclosed
EP-0786455-A1 IMIDAZOLE DERIVATIVE SHIONOGI & CO., LTD. (JP) 1997-07-30 EP disclosed