SCHEMBL6977345

SCHEMBL6977345

COc1ccc2nccc(C[C@H](O)CC3CCNCC3)c2c1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.51
NCF1 P14598 1/20 0.47
MTNR1A P48039 3/20 0.45
MTNR1B P49286 3/20 0.45
KCNH2 Q12809 3/20 0.42
LMNA P02545 1/20 0.41
DYRK3 O43781 1/20 0.41
CLK1 P49759 1/20 0.41
CLK2 P49760 1/20 0.41
CLK3 P49761 1/20 0.41
DYRK1A Q13627 1/20 0.41
DYRK2 Q92630 1/20 0.41
CLK4 Q9HAZ1 1/20 0.41
DYRK4 Q9NR20 1/20 0.41
DYRK1B Q9Y463 1/20 0.41
TDP1 Q9NUW8 1/20 0.41
KDM4E B2RXH2 3/20 0.40
CYP2D6 P10635 3/20 0.40
ALDH1A1 P00352 2/20 0.40
HPGD P15428 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977344 1.00 ROCK2 (0.51) ROCK2NCF1MTNR1AMTNR1BKCNH2
SCHEMBL6977351 1.00 ROCK2 (0.51) ROCK2NCF1MTNR1AMTNR1BKCNH2
SCHEMBL6971430 0.83 NCF1 (0.49) NCF1KCNH2TDP1KDM4ECYP2D6
SCHEMBL6971434 0.83 NCF1 (0.49) NCF1KCNH2TDP1KDM4ECYP2D6
SCHEMBL6971431 0.83 NCF1 (0.49) NCF1KCNH2TDP1KDM4ECYP2D6
SCHEMBL10953793 0.81 KCNH2 (0.59) NCF1MTNR1AMTNR1BKCNH2
Hydrochloric Acid SCHEMBL10953152 0.80 KCNH2 (0.58) NCF1MTNR1AMTNR1BKCNH2TDP1
SCHEMBL6977177 0.80 CCR8 (0.53) ROCK2MTNR1AMTNR1BKCNH2KDM4E
SCHEMBL6977170 0.80 CCR8 (0.53) ROCK2MTNR1AMTNR1BKCNH2KDM4E
SCHEMBL6977174 0.80 CCR8 (0.53) ROCK2MTNR1AMTNR1BKCNH2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1051413-B1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2003-06-04 EP disclosed
EP-1051413-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 2000-11-15 EP disclosed
WO-1999037635-A1 QUINOLINE DERIVATIVES AS ANTIBACTERIALS SMITHKLINE BEECHAM PLC (GB) 1999-07-29 WO disclosed