SCHEMBL6977429

SCHEMBL6977429

COC(=O)c1ccccc1CCC1CCCCN=C1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.46
LMNA P02545 1/20 0.46
KDM4E B2RXH2 5/20 0.40
HSD17B10 Q99714 2/20 0.40
HPGD P15428 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
TSHR P16473 2/20 0.38
DRD1 P21728 1/20 0.37
HRH2 P25021 1/20 0.37
HTR2A P28223 1/20 0.37
HTR2C P28335 1/20 0.37
OPRK1 P41145 1/20 0.37
HTR2B P41595 1/20 0.37
KCNH2 Q12809 1/20 0.37
RECQL P46063 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
RIPK1 Q13546 1/20 0.36
ATM Q13315 1/20 0.36
ADRA1D P25100 1/20 0.36
ADRA1A P35348 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21180879 0.78 ALDH1A1 (0.57) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL6980114 0.76 ALDH1A1 (0.47) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL6972034 0.75 ALDH1A1 (0.46) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL6976786 0.73 ALDH1A1 (0.46) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL10360804 0.71 ALDH1A1 (0.77) ALDH1A1LMNAKDM4EHSD17B10TSHR
SCHEMBL6979274 0.70 STS (0.42) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL6979271 0.70 STS (0.42) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL6979269 0.70 STS (0.42) ALDH1A1LMNAKDM4EHSD17B10HPGD
SCHEMBL19515023 0.70 ALDH1A1 (0.55) ALDH1A1LMNAKDM4EHSD17B10HPGD
Hydrochloric Acid SCHEMBL19515032 0.69 ALDH1A1 (0.53) ALDH1A1LMNAKDM4EHSD17B10HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6043261-A TREATMENT OF INFLAMMATORY CONDITIONS AFFECTING THE JOINTS, FOR EXAMPLE ARTHRITIS, INFLAMMATORY BOWEL DISEASE, CARDIOVASCULAR ISCHEMIA, DIABETES, HYPERALGESIA, CEREBRAL ISCHEMIA, THROMBOTIC STROKE, GLOBAL ISCHEMIA, NERVOUS SYSTEM DISORDERS G. D. SEARLE & CO. (US) 2000-03-28 US disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
US-5883251-A ENZYME INHIBITORS G. D. SEARLE & CO. (US) 1999-03-16 US disclosed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO disclosed