SCHEMBL6977552

SCHEMBL6977552

O=C(Nc1ccc(F)cc1)C(F)Cl

nearest known ligand 0.53

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.53
MEN1 O00255 6/20 0.53
KMT2A Q03164 6/20 0.53
CYP1A2 P05177 1/20 0.53
CYP2C9 P11712 1/20 0.53
CYP2C19 P33261 1/20 0.53
MAPT P10636 2/20 0.49
RECQL P46063 1/20 0.49
TGM2 P21980 1/20 0.48
SMN1; SMN2 Q16637 4/20 0.47
NPC1 O15118 3/20 0.47
RAB9A P51151 3/20 0.47
HTT P42858 3/20 0.47
POLB P06746 3/20 0.47
TAAR1 Q96RJ0 1/20 0.47
GAA P10253 1/20 0.47
PTPN1 P18031 1/20 0.47
MITF O75030 1/20 0.46
HPGD P15428 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30513730 0.83 ALDH1A1 (0.57) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL7939406 0.82 MEN1 (0.61) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL5417260 0.78 MEN1 (0.51) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL10819622 0.78 KMT2A (0.80) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL29522603 0.77 KMT2A (0.58) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL9470930 0.77 MAPT (0.71) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL27046122 0.75 EPHX2 (0.65) ALDH1A1MEN1KMT2AMAPTSMN1; SMN2
SCHEMBL11734595 0.74 KMT2A (0.60) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL8274716 0.74 TAAR1 (0.64) ALDH1A1MEN1KMT2ACYP1A2CYP2C9
SCHEMBL29521778 0.74 ALDH1A1 (0.52) ALDH1A1MEN1KMT2ACYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1077947-B1 NOVEL 1,5 AND 3-O-SUBSTITUTED 1H-INDAZOLES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY, IMMUNO-MODULATING AND NEURO-PROTECTIVE EFFECT, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS DRESDEN ARZNEIMITTEL (DE) 2003-09-03 EP disclosed
EP-1077947-A1 NOVEL 1,5 AND 3-O-SUBSTITUTED 1H-INDAZOLES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY, IMMUNO-MODULATING AND NEURO-PROTECTIVE EFFECT, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS ARZNEIMITTELWERK DRESDEN GMBH (DE) 2001-02-28 EP disclosed
US-6166023-A 1,5- and 3-O-substituted 1H-indazoles having anti-asthmatic, anti-allergic, anti-inflammatory, immunomodulating and neuroprotective action, process for their preparation and their use as medicaments ARZNEIMITTELWERK DRESDEN GMBH (DE) 2000-12-26 US disclosed
WO-1999058503-A1 NOVEL 1,5 AND 3-O-SUBSTITUTED 1H-INDAZOLES WITH ANTI-ASTHMATIC, ANTI-ALLERGIC, ANTI-INFLAMMATORY, IMMUNO-MODULATING AND NEURO-PROTECTIVE EFFECT, METHOD FOR THE PRODUCTION AND USE THEREOF AS MEDICAMENTS ARZNEIMITTELWERK DRESDEN GMBH (DE) 1999-11-18 WO disclosed