SCHEMBL6977841

SCHEMBL6977841

O=C(NNCc1ccccc1)C1CC(SC(c2ccccc2)(c2ccccc2)c2ccccc2)CN1S(=O)(=O)c1ccc2ccccc2c1

nearest known ligand 0.43

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CCR4 P51679 6/20 0.43
MME P08473 2/20 0.42
ACE P12821 2/20 0.42
ECE1 P42892 2/20 0.42
MMP9 P14780 1/20 0.41
CAPN1 P07384 1/20 0.40
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
EIF2AK3 Q9NZJ5 1/20 0.38
HCRTR1 O43613 1/20 0.38
HCRTR2 O43614 1/20 0.38
MMP1 P03956 4/20 0.37
ADAM17 P78536 3/20 0.37
AKR1C3 P42330 3/20 0.37
AKR1C1 Q04828 1/20 0.37
MMP2 P08253 1/20 0.37
MMP3 P08254 1/20 0.37
MMP7 P09237 1/20 0.37
MMP13 P45452 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5723069 1.00 CCR4 (0.43) CCR4MMEACEECE1MMP9
SCHEMBL5723096 0.88 TRPA1 (0.43) CCR4MMEACEECE1LMNA
SCHEMBL7146134 0.86 LMNA (0.51) CCR4MMEACEECE1MMP9
SCHEMBL5723986 0.86 MME (0.47) CCR4MMEACEECE1MMP9
SCHEMBL5723228 0.86 MME (0.47) CCR4MMEACEECE1MMP9
SCHEMBL6978080 0.84 AKR1C3 (0.47) CCR4MMEACEECE1LMNA
SCHEMBL5402095 0.84 AKR1C3 (0.47) CCR4MMEACEECE1LMNA
SCHEMBL5723508 0.84 HDAC3 (0.41) CCR4MMEACEECE1MMP9
SCHEMBL5723585 0.83 ECE1 (0.59) CCR4MMEACEECE1MMP9
SCHEMBL6968343 0.82 MME (0.43) CCR4MMEACEECE1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317428-A1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2003-06-11 EP disclosed
WO-2002006224-A1 PYRROLIDINE-2-CARBOXYLIC ACID HYDRAZIDE DERIVATIVES FOR USE AS METALLOPROTEASE INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed