SCHEMBL6978153

SCHEMBL6978153

CC(C)(C)N[C@@H]1C[C@@H](COCc2ccccc2)N(C(=O)O)C1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AGTR2 P50052 2/20 0.41
NR1D1 P20393 1/20 0.39
OPRM1 P35372 1/20 0.37
OPRD1 P41143 1/20 0.37
OPRK1 P41145 1/20 0.37
ABHD6 Q9BV23 1/20 0.36
DAGLA Q9Y4D2 1/20 0.36
EPHX2 P34913 1/20 0.35
RIPK1 Q13546 1/20 0.35
DPP4 P27487 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
FKBP1A P62942 1/20 0.35
CTSL P07711 1/20 0.34
CTSB P07858 1/20 0.34
CTSK P43235 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22555190 0.79 AGTR2 (0.46) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL6975692 0.79 AGTR2 (0.46) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL4297034 0.79 AGTR2 (0.46) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL6978115 0.78 AGTR2 (0.46) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL4294638 0.78 AGTR2 (0.46) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL21752301 0.76 AGTR2 (0.39) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL4303290 0.76 AGTR2 (0.39) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL22555092 0.75 AGTR2 (0.48) AGTR2NR1D1OPRM1OPRD1OPRK1
SCHEMBL20974188 0.74 CA12 (0.38) KMT2A
SCHEMBL20479729 0.74 ALDH1A1 (0.50) DPP4CTSLCTSBCTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1100797-B1 HETEROCYCLIC COMPOUNDS AS INHIBITORS OF ROTAMASE ENZYMES PFIZER LTD (GB) 2003-02-26 EP disclosed