SCHEMBL6979877

SCHEMBL6979877

Cc1ccccc1-c1cc(N2CCSCC2)nc(C)c1C(N)=O

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKDC P78527 1/20 0.37
ALDH1A1 P00352 4/20 0.36
HPGD P15428 4/20 0.36
POLB P06746 1/20 0.36
ALOX12 P18054 1/20 0.36
IKBKB O14920 4/20 0.36
PLA2G7 Q13093 1/20 0.36
TACR1 P25103 3/20 0.36
TDP1 Q9NUW8 2/20 0.35
KDM4E B2RXH2 2/20 0.34
HSD17B10 Q99714 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
USP2 O75604 1/20 0.34
LMNA P02545 1/20 0.34
TSHR P16473 1/20 0.34
MAPK1 P28482 1/20 0.34
CYP1A2 P05177 1/20 0.34
GBA1 P04062 4/20 0.34
MAPT P10636 1/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1399406 0.76 MAPT (0.49) ALDH1A1HPGDIKBKBTACR1KDM4E
SCHEMBL4374050 0.72 CYP1A2 (0.43) ALDH1A1TACR1TSHRCYP1A2
SCHEMBL30572211 0.71 NNMT (0.45) ALDH1A1HPGDIKBKBKDM4EHSD17B10
SCHEMBL905377 0.70 TACR1 (0.45) TACR1CYP1A2
SCHEMBL4374612 0.69 TACR1 (0.43) ALDH1A1TACR1MAPT
SCHEMBL4374064 0.68 CYP1A2 (0.41) ALDH1A1TACR1HSD17B10TSHRCYP1A2
SCHEMBL17476483 0.67 ALDH1A1 (0.43) PRKDCALDH1A1HPGDIKBKBTACR1
SCHEMBL23277178 0.67 IKBKB (0.56) POLBIKBKBKDM4E
SCHEMBL3095284 0.67 IKBKB (0.56) ALDH1A1HPGDPOLBIKBKBKDM4E
SCHEMBL27473965 0.67 MKNK1 (0.46) ALDH1A1IKBKBPLA2G7TDP1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303490-A1 N-OXIDES AS NK1 RECEPTOR ANTAGONIST PRODRUGS OF 4-PHENYL-PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2003-04-23 EP disclosed
WO-2002006236-A1 N-OXIDES AS NK1 RECEPTOR ANTAGONIST PRODRUGS OF 4-PHENYL-PYRIDINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2002-01-24 WO disclosed