SCHEMBL6980039

SCHEMBL6980039

O=C1CCCCC(CCc2ccncc2)N1

nearest known ligand 0.43

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 2/20 0.43
GAA P10253 1/20 0.43
MMP13 P45452 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
HSD17B10 Q99714 1/20 0.37
CTSD P07339 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6976834 0.82 GAA (0.37) CYP19A1GAAMMP13RAB9ASMN1; SMN2
Hydrochloric Acid SCHEMBL6978274 0.81 GAA (0.36) CYP19A1GAAMMP13RAB9ASMN1; SMN2
SCHEMBL5963304 0.80 CTSD (0.43) CTSD
SCHEMBL6977505 0.77 NR1H4 (0.36) CTSD
SCHEMBL13336109 0.77 DAO (0.42)
SCHEMBL6979908 0.77 CTSD (0.43) CTSD
SCHEMBL6969464 0.76 HSD17B10 (0.40) RAB9ASMN1; SMN2HSD17B10
SCHEMBL6978291 0.75 CTSD (0.45) CTSD
SCHEMBL22652854 0.75 HRH3 (0.55)
SCHEMBL29742940 0.75 KMT2A (0.35) CTSD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
EP-0821674-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-02-04 EP disclosed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO disclosed