SCHEMBL6969464

SCHEMBL6969464

O=C1CCCCC(CCc2ccccn2)N1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B10 Q99714 1/20 0.40
DDB1 Q16531 1/20 0.40
CRBN Q96SW2 1/20 0.40
HRH3 Q9Y5N1 3/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
HRH1 P35367 1/20 0.38
CYP1A2 P05177 1/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
DPP7 Q9UHL4 1/20 0.38
RECQL P46063 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
PDCD1 Q15116 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978536 0.84 HRH3 (0.39) HRH3HPGDNPC1RAB9ASMN1; SMN2
SCHEMBL6980039 0.76 CYP19A1 (0.43) HSD17B10RAB9ASMN1; SMN2
SCHEMBL6975941 0.76 KDM4E (0.49) HSD17B10HRH3HPGDNPC1RAB9A
SCHEMBL2136372 0.76 CRBN (0.44) DDB1CRBNSMN1; SMN2MEN1KMT2A
SCHEMBL6978540 0.75 HRH3 (0.41) HSD17B10HRH3NPC1RAB9ASMN1; SMN2
SCHEMBL13009896 0.74 LMNA (0.36) CYP1A2CYP3A4CYP2D6CYP2C9CYP2C19
SCHEMBL5963304 0.74 CTSD (0.43)
SCHEMBL6979908 0.73 CTSD (0.43)
SCHEMBL6978291 0.72 CTSD (0.45)
SCHEMBL6850513 0.71 HPGD (0.57) HSD17B10HRH3HPGDNPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0821674-B1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS SEARLE & CO (US) 2003-08-06 EP disclosed
US-6011028-A Cyclic amidino agents useful as nitric oxide synthase inhibitors G.D. SEARLE & CO. (US) 2000-01-04 US disclosed
EP-0821674-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1998-02-04 EP disclosed
WO-1996033175-A1 CYCLIC AMIDINO AGENTS USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS G.D. SEARLE & CO. (US) 1996-10-24 WO disclosed