SCHEMBL6980329

SCHEMBL6980329

COc1ccc2c(c1)OC(c1c(C)ccc(S(=O)(=O)O)c1C)CN2C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
STS P08842 2/20 0.35
MMP1 P03956 2/20 0.35
MMP9 P14780 2/20 0.35
MMP3 P08254 1/20 0.35
MMP7 P09237 1/20 0.35
RORC P51449 3/20 0.34
MMP13 P45452 1/20 0.34
ALDH1A1 P00352 3/20 0.33
MEN1 O00255 2/20 0.33
KMT2A Q03164 2/20 0.33
NFKB1 P19838 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
NOTUM Q6P988 1/20 0.33
CYP3A4 P08684 2/20 0.33
POLB P06746 1/20 0.33
CYP2C9 P11712 1/20 0.33
SIRT3 Q9NTG7 1/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
PKM P14618 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977474 0.76 MAPT (0.44) RORCALDH1A1NFKB1NFKB2RELA
SCHEMBL3359225 0.74 KMT2A (0.46) STSRORCALDH1A1MEN1KMT2A
SCHEMBL8662867 0.74 FFAR1 (0.39)
SCHEMBL8666860 0.74 FFAR1 (0.39)
SCHEMBL7822268 0.73 ALDH1A1 (0.39) STSMMP1MMP9MMP3MMP7
SCHEMBL3353116 0.72 ALDH1A1 (0.51) ALDH1A1MEN1KMT2ACYP3A4POLB
SCHEMBL6980332 0.69 EPHX2 (0.38) RORCALDH1A1MEN1KMT2ANOTUM
SCHEMBL31371813 0.66 USP30 (0.43) STSALDH1A1MEN1KMT2ANFKB1
SCHEMBL5389996 0.66 NOTUM (0.68) KMT2ANOTUMSMN1; SMN2GPR119
SCHEMBL23878317 0.65 MEN1 (0.41) STSMMP13ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1140925-B1 (3,4 DIHYDRO-2H-BENZO[1,4] OXAZINYL-METHYL)- 3-(1H-INDOL-3- YL)-ALKYL -AMINES WYETH CORP (US) 2003-04-23 EP disclosed
US-6313114-B1 ANTIDEPRESSANTS AMERICAN HOME PRODUCTS CORP 2001-11-06 US disclosed
EP-1140925-A1 (3,4 DIHYDRO-2H-BENZO[1,4] OXAZINYL-METHYL)- 3-(1H-INDOL-3- YL)-ALKYL -AMINES AMERICAN HOME PRODUCTS CORPORATION (US) 2001-10-10 EP disclosed
WO-2000040580-A1 3,4-DIHYDRO-2H-BENZO[1,4]OXAZINYL-METHYL[3-(1H-INDOL-3-YL)-ALKYL]-AMINES AMERICAN HOME PRODUCTS CORPORATION (US) 2000-07-13 WO disclosed