SCHEMBL6980488

SCHEMBL6980488

CS(=O)(=O)c1ccc(-n2nc(C(F)F)cc2-c2nc3ccc(Cl)cc3s2)cc1

nearest known ligand 0.51

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 15/20 0.51
PTGS1 P23219 8/20 0.51
CCNE1 P24864 1/20 0.41
CDK2 P24941 1/20 0.41
CDK5 Q00535 1/20 0.41
CDK5R1 Q15078 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978991 0.90 PTGS2 (0.64) PTGS2PTGS1CCNE1CDK2CDK5
SCHEMBL6974226 0.90 PTGS2 (0.53) PTGS2PTGS1CCNE1CDK2CDK5
SCHEMBL6972326 0.89 PTGS2 (0.48) PTGS2PTGS1CCNE1CDK2CDK5
SCHEMBL6978365 0.87 PTGS2 (0.50) PTGS2PTGS1
SCHEMBL6981308 0.87 PTGS1 (0.54) PTGS2PTGS1
SCHEMBL6983224 0.85 PTGS2 (0.55) PTGS2PTGS1
SCHEMBL6982997 0.83 PTGS2 (0.45) PTGS2PTGS1
SCHEMBL6979695 0.83 PTGS2 (0.48) PTGS2PTGS1
SCHEMBL6972090 0.81 PTGS2 (0.66) PTGS2PTGS1CCNE1CDK2CDK5
SCHEMBL6982484 0.79 PTGS2 (0.56) PTGS2PTGS1CCNE1CDK2CDK5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed