SCHEMBL6981658

SCHEMBL6981658

NS(=O)(=O)c1ccc(-n2nc(C(F)F)cc2-c2nc3cccc(Cl)c3s2)cc1

nearest known ligand 0.61

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 18/20 0.61
PTGS1 P23219 13/20 0.61
ABCB11 O95342 1/20 0.48
ALDH1A1 P00352 1/20 0.48
PDPK1 O15530 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6977045 0.90 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6975857 0.89 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6981121 0.85 PTGS2 (0.64) PTGS2PTGS1PDPK1
SCHEMBL6972333 0.85 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6978991 0.82 PTGS2 (0.64) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL6982413 0.80 PTGS2 (0.45) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6980897 0.79 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6982484 0.79 PTGS2 (0.56) PTGS2PTGS1ABCB11ALDH1A1
SCHEMBL6972090 0.79 PTGS2 (0.66) PTGS2PTGS1ABCB11ALDH1A1PDPK1
SCHEMBL6980516 0.78 PTGS2 (0.58) PTGS2PTGS1ABCB11ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1006114-B1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM GRELAN PHARMACEUTICAL CO (JP) 2003-01-22 EP disclosed
US-6136831-A ANTIINFLAMMATORY AGENTS, GASTROINTESTINAL AGENTS, ENZYME INHIBITORS GRELAN PHARMACEUTICAL CO., LTD. (JP) 2000-10-24 US disclosed
EP-1006114-A1 PYRAZOLE DERIVATIVES AND COX INHIBITORS CONTAINING THEM Grelan Pharmaceutical Co., Ltd. (JP) 2000-06-07 EP disclosed