SCHEMBL6982022

SCHEMBL6982022

CCc1nnc(CCCOc2c(C)cc(-c3noc(C)n3)cc2C)s1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
S1PR1 P21453 13/20 0.38
S1PR3 Q99500 11/20 0.38
L3MBTL1 Q9Y468 1/20 0.37
SCARB1 Q8WTV0 1/20 0.35
ACACB O00763 1/20 0.33
ACACA Q13085 1/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6974407 0.91 NR1I2 (0.47) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL6976401 0.86 NR1I2 (0.45) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL9090154 0.85 NR1I2 (0.46) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL8687271 0.83 NR1I2 (0.46) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL8555393 0.82 NR1I2 (0.45) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL8912937 0.81 NR1I2 (0.47) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL9087864 0.80 NR1I2 (0.47) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL9205929 0.79 NR1I2 (0.57) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL8670645 0.77 CYP3A4 (0.48) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL8553518 0.77 NR1I2 (0.49) NR1I2CYP3A4CYP2D6S1PR1L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0759755-B1 Thiadiazolylalkoxyphenyl derivatives, their preparation and their use anti-picornaviral agents SANOFI SYNTHELABO (FR) 2003-08-13 EP disclosed
US-5650419-A Thiadiazoles and their use as antipicornaviral agents SANOFI, S.A. 1997-07-22 US disclosed
EP-0759755-A4 THIADIAZOLES AND THEIR USE AS ANTIPICORNAVIRAL AGENTS SANOFI WINTHROP INC (US) 1997-05-07 EP disclosed
EP-0759755-A1 Thiadiazolylalkoxyphenyl derivatives, their preparation and their use anti-picornaviral agents SANOFI WINTHROP, INC. (US) 1997-03-05 EP disclosed
US-5567719-A Thiadiazoles and their use as antipicornaviral agents STERLING WINTHROP, INC. (US) 1996-10-22 US disclosed
WO-1995031198-A1 THIADIAZOLES AND THEIR USE AS ANTIPICORNAVIRAL AGENTS SANOFI WINTHROP, INC. (US) 1995-11-23 WO disclosed
US-5453433-A Viricides; antiseptics to decontaminate polio, rhino and coxsackie viruses STERLING WINTHROP INC. (US) 1995-09-26 US disclosed