SCHEMBL8912937

SCHEMBL8912937

Cc1nsc(CCCOc2c(C)cc(-c3noc(C)n3)cc2C)n1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR1I2 O75469 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2D6 P10635 1/20 0.47
L3MBTL1 Q9Y468 2/20 0.37
S1PR1 P21453 6/20 0.33
S1PR3 Q99500 5/20 0.33
CA12 O43570 1/20 0.33
CA1 P00915 1/20 0.33
CA2 P00918 1/20 0.33
CA9 Q16790 1/20 0.33
TDP1 Q9NUW8 2/20 0.32
HDAC1 Q13547 1/20 0.31
HDAC8 Q9BY41 1/20 0.31
HDAC6 Q9UBN7 1/20 0.31
AOC3 Q16853 2/20 0.31
SCARB1 Q8WTV0 1/20 0.31
MAOA P21397 1/20 0.31
MAOB P27338 1/20 0.31
LMNA P02545 1/20 0.31
MAPT P10636 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6983983 0.87 NR1I2 (0.46) NR1I2CYP3A4CYP2D6S1PR1S1PR3
SCHEMBL6974407 0.81 NR1I2 (0.47) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL6982022 0.81 NR1I2 (0.47) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL8687271 0.81 NR1I2 (0.46) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL8553518 0.80 NR1I2 (0.49) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL9090154 0.78 NR1I2 (0.46) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL9087864 0.78 NR1I2 (0.47) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL8670645 0.77 CYP3A4 (0.48) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL8555393 0.77 NR1I2 (0.45) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1
SCHEMBL9200266 0.77 NR1I2 (0.73) NR1I2CYP3A4CYP2D6L3MBTL1S1PR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5650419-A Thiadiazoles and their use as antipicornaviral agents SANOFI, S.A. 1997-07-22 US disclosed
US-5567719-A Thiadiazoles and their use as antipicornaviral agents STERLING WINTHROP, INC. (US) 1996-10-22 US disclosed
US-5453433-A Viricides; antiseptics to decontaminate polio, rhino and coxsackie viruses STERLING WINTHROP INC. (US) 1995-09-26 US disclosed