SCHEMBL6982224

SCHEMBL6982224

O=C(c1cn(Cc2c[nH]cn2)cc1-c1ccc2c3c(cccc13)CC2)N1CCOCC1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.53
ALDH1A1 P00352 3/20 0.53
HSD17B10 Q99714 2/20 0.53
MEN1 O00255 1/20 0.53
HPGD P15428 1/20 0.53
KMT2A Q03164 1/20 0.53
FNTA P49354 8/20 0.51
FNTB P49356 8/20 0.51
PGGT1B P53609 2/20 0.40
MAPK1 P28482 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.38
USP2 O75604 1/20 0.36
CYP3A4 P08684 1/20 0.35
HRH3 Q9Y5N1 1/20 0.35
PLAUR Q03405 1/20 0.34
CNR1 P21554 1/20 0.34
CNR2 P34972 1/20 0.34
ALOX5AP P20292 1/20 0.34
FEN1 P39748 1/20 0.34
MAPT P10636 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6975190 0.86 FNTA (0.69) ALDH1A1MEN1KMT2AFNTAFNTB
SCHEMBL6977285 0.82 FNTA (0.53) KDM4EALDH1A1HSD17B10MEN1HPGD
SCHEMBL6977393 0.78 FNTA (0.57) KDM4EALDH1A1HSD17B10FNTAFNTB
SCHEMBL6975380 0.77 FNTA (0.56) KDM4EFNTAFNTBPGGT1BCYP3A4
SCHEMBL6982604 0.77 FNTA (0.61) ALDH1A1MEN1KMT2AFNTAFNTB
SCHEMBL6982870 0.77 FNTA (0.68) KDM4EFNTAFNTBPGGT1BCYP3A4
SCHEMBL6979480 0.76 FNTA (0.57) FNTAFNTBPGGT1BCYP3A4PLAUR
SCHEMBL6982219 0.74 FNTA (0.57) FNTAFNTBPGGT1BCYP3A4
SCHEMBL6984228 0.74 FNTA (0.55) KDM4EFNTAFNTBPGGT1BCYP3A4
SCHEMBL6980781 0.72 FNTA (0.52) FNTAFNTBPGGT1BCYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP claimed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US claimed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof FNTA, FNTB, FDPS KDM4E 2589/4885ALDH1A1 646/4885HSD17B10 661/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.