SCHEMBL6983095

SCHEMBL6983095

O=S(=O)(Nc1ccc2c(c1)CCCN2)c1cccc2ccccc12

nearest known ligand 0.51

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.51
ALDH1A1 P00352 1/20 0.49
HTT P42858 1/20 0.49
PFKFB3 Q16875 1/20 0.49
TSHR P16473 1/20 0.48
PGR P06401 1/20 0.48
PARP1 P09874 1/20 0.48
HDAC1 Q13547 1/20 0.47
HTR6 P50406 8/20 0.47
GHSR Q92847 2/20 0.47
PTPN2 P17706 1/20 0.45
PTPN1 P18031 1/20 0.45
PTPN5 P54829 1/20 0.45
RORA P35398 1/20 0.45
RORC P51449 1/20 0.45
NR1H2 P55055 1/20 0.45
NR1H4 Q96RI1 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6980011 0.83 BRD4 (0.58) BRD4ALDH1A1PTPN2PTPN1PTPN5
SCHEMBL6984820 0.80 HTR6 (0.61) BRD4ALDH1A1HTR6
SCHEMBL6976538 0.80 PKM (0.65) BRD4ALDH1A1HTTPGRHTR6
SCHEMBL6985547 0.78 HTR6 (0.41) BRD4HDAC1HTR6
SCHEMBL4709118 0.78 HTR6 (0.55) BRD4ALDH1A1HTTPFKFB3TSHR
SCHEMBL10238657 0.78 HTR6 (0.55) BRD4ALDH1A1HTTPFKFB3TSHR
Hydrochloric Acid SCHEMBL9960412 0.77 HTR6 (0.54) BRD4ALDH1A1HTTPFKFB3TSHR
Hydrochloric Acid SCHEMBL3156784 0.77 HTR6 (0.54) BRD4ALDH1A1HTTPFKFB3TSHR
SCHEMBL31681377 0.76 EIF2AK2 (0.54) BRD4ALDH1A1HTR6GHSR
SCHEMBL6983098 0.76 HCRTR1 (0.43) ALDH1A1TSHRPGRHTR6GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed