SCHEMBL6983374

SCHEMBL6983374

COC(=O)c1sc(C(Cc2ccc(Cl)cc2)c2cnc[nH]2)nc1-c1cccc2ccccc12

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 2/20 0.38
GAA P10253 1/20 0.38
KMT2A Q03164 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ADRA2A P08913 6/20 0.37
ADRA2B P18089 6/20 0.37
ADRA2C P18825 6/20 0.37
CPA1 P15085 1/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.36
ADRA1A P35348 4/20 0.35
ADRA1D P25100 3/20 0.35
ADRA1B P35368 3/20 0.35
FNTA P49354 2/20 0.35
FNTB P49356 2/20 0.35
PGGT1B P53609 1/20 0.35
CPB2 Q96IY4 1/20 0.34
S1PR1 P21453 1/20 0.34
MAPT P10636 2/20 0.33
LMNA P02545 1/20 0.33
HPGD P15428 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6978781 0.87 ADRA2A (0.37) KDM4EGAAKMT2ANPSR1ADRA2A
SCHEMBL6981192 0.83 FNTA (0.46) KMT2AFNTAFNTBPGGT1B
SCHEMBL6923536 0.77 HTR2C (0.44) KMT2AADRA2AADRA2BADRA2CCPA1
SCHEMBL6980881 0.73 FNTA (0.46) GAAKMT2ANPSR1FNTAFNTB
SCHEMBL6983372 0.70 FNTA (0.48) KDM4EGAAKMT2ANPSR1FNTA
SCHEMBL6973808 0.68 FNTA (0.42) ADRA2AADRA2BADRA2CFNTAFNTB
SCHEMBL6984368 0.65 FNTA (0.54) KDM4EGAAKMT2AFNTAFNTB
SCHEMBL6610055 0.64 ADRA2A (0.38) ADRA2AADRA2BADRA2CCPA1ADRA1A
SCHEMBL6599134 0.63 FNTA (0.37) KDM4EADRA2AADRA2BADRA2CADRA1A
SCHEMBL8764039 0.61 CPA1 (0.72) CPA1CPB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP claimed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US claimed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US claimed
EP-1045846-B1 IMIDAZOLE DERIVATIVES HAVING AN INHIBITORY ACTIVITY FOR FARNESYL TRANSFERASE AND PROCESS FOR PREPARATION THEREOF LG CHEMICAL LTD (KR) 2003-05-02 EP disclosed
US-6518429-B2 Anticancer agents, treating restenosis, atherosclerosis and hepatitis virus LG CHEMICAL, LTD. (KR) 2003-02-11 US disclosed
US-6472526-B1 SHOWS AN INHIBITORY ACTIVITY AGAINST FARNESYL TRANSFERASE OR PHARMACEUTICALLY ACCEPTABLE SALTS OR ISOMERS THEREOF, IN PHARMACEUTICAL COMPOSITION AND INTERMEDIATES LG CHEMICAL LTD. (KR) 2002-10-29 US disclosed
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof LG CHEMICAL LTD. 2002-09-26 US disclosed
US-6268363-B1 ANTITUMOR LG CHEMICAL LTD. (KR) 2001-07-31 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20020137769-A1 Imidazole derivatives having an inhibitory activity for farnesyl transferase and process for preparation thereof FNTA, FNTB, FDPS KDM4E 2589/4885GAA 470/4885KMT2A 3370/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.