SCHEMBL6983930

SCHEMBL6983930

Cc1c(C)c2c(c(C)c1N)CC(C)(CN1CCC(OC(c3ccccc3)c3ccccc3)CC1)O2

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 3/20 0.43
ADRA2A P08913 3/20 0.43
CHRM1 P11229 3/20 0.43
DRD1 P21728 3/20 0.43
SLC6A2 P23975 3/20 0.43
ADRA1A P35348 3/20 0.43
DRD3 P35462 3/20 0.43
SLC6A3 Q01959 3/20 0.43
KCNH2 Q12809 3/20 0.43
HTR1A P08908 2/20 0.43
OPRM1 P35372 2/20 0.43
CYP2D6 P10635 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43
MAPK1 P28482 1/20 0.42
BCHE P06276 8/20 0.37
GRM5 P41594 1/20 0.37
GRM7 Q14831 1/20 0.37
GRM3 Q14832 1/20 0.37
HPGDS O60760 1/20 0.37
CHRM4 P08173 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Oxalic Acid SCHEMBL6980644 0.95 GRM5 (0.42) CHRM2ADRA2ACHRM1DRD1SLC6A2
SCHEMBL6979549 0.91 CHRM2 (0.44) CHRM2ADRA2ACHRM1DRD1SLC6A2
Oxalic Acid SCHEMBL6985362 0.88 BCHE (0.40) SLC6A2SLC6A3BCHEGRM5GRM7
SCHEMBL6976596 0.87 KCNA3 (0.41)
Oxalic Acid SCHEMBL6983672 0.87 BCHE (0.43) CHRM2ADRA2ACHRM1DRD1SLC6A2
SCHEMBL6980205 0.83 CARM1 (0.43) OPRM1HRH3BCHESIGMAR1
Oxalic Acid SCHEMBL6977629 0.83 SLC6A4 (0.39) SLC6A2SLC6A3SLC6A4
Hydrochloric Acid SCHEMBL6984798 0.83 SMN1; SMN2 (0.43) CHRM2ADRA2ACHRM1DRD1SLC6A2
SCHEMBL6976347 0.83 CHRM1 (0.32) CHRM1SLC6A2SLC6A4
SCHEMBL6983686 0.83 CHRM1 (0.32) CHRM1SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0923575-B1 CYCLIC ETHER COMPOUNDS AS SODIUM CHANNEL MODULATORS TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2003-03-12 EP disclosed
US-6172085-B1 CENTRAL NERVOUS SYSTEM AND PSYCHOLOGICAL DISORDERS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 2001-01-09 US disclosed