SCHEMBL6984152

SCHEMBL6984152

COc1ccc(C[C@@H](N(O)C=O)S(=O)(=O)Cc2ccc3occc3c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTR1B P28222 4/20 0.38
CA2 P00918 7/20 0.38
CA12 O43570 4/20 0.37
LDHA P00338 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.35
MRGPRX4 Q96LA9 1/20 0.35
MMP1 P03956 1/20 0.35
MMP9 P14780 1/20 0.35
MMP13 P45452 1/20 0.35
ADAM17 P78536 1/20 0.35
POLB P06746 1/20 0.34
CTNNB1 P35222 1/20 0.34
WNT3A P56704 1/20 0.34
TAS1R3 Q7RTX0 1/20 0.34
TAS1R1 Q7RTX1 1/20 0.34
PIN1 Q13526 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6399534 0.81 HTR1B (0.36) HTR1BCA2CA12SIRT2MMP9
SCHEMBL6399540 0.81 HTR1B (0.36) HTR1BCA2CA12SIRT2MMP9
SCHEMBL6605359 0.77 CA2 (0.39) HTR1BCA2CA12SIRT2MRGPRX4
SCHEMBL6400527 0.69 KMT2A (0.34) CA2MRGPRX4POLBPIN1
SCHEMBL6404097 0.69 MMP2 (0.39) HTR1BCA2CA12MRGPRX4MMP9
SCHEMBL6400988 0.69 MMP2 (0.39) HTR1BCA2CA12MRGPRX4MMP9
SCHEMBL12773195 0.67 SMN1; SMN2 (0.48) HTR1BPOLB
SCHEMBL15979957 0.64 CTNNB1 (0.72) HTR1BMMP1CTNNB1WNT3ATAS1R3
SCHEMBL826624 0.64 CYP2A6 (0.55) CA2CA12
SCHEMBL463181 0.64 CA2 (0.48) HTR1BCA2CA12CTNNB1WNT3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289980-A1 BICYCLYL OR HETEROBICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED N-HYDROXYFORMAMIDES SMITHKLINE BEECHAM PLC (GB) 2003-03-12 EP disclosed
WO-2001090100-A1 BICYCLYL OR HETEROBICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED N-HYDROXYFORMAMIDES SMITHKLINE BEECHAM P.L.C. (GB) 2001-11-29 WO disclosed