SCHEMBL6984478

SCHEMBL6984478

CCOC(=O)CN(c1ccc2c(c1)CCCN2C(=O)CCc1ccc(C(=N)NC(=O)OC)cc1)S(=O)(=O)c1cccc2cccnc12

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
F2 P00734 5/20 0.42
ALDH1A1 P00352 4/20 0.41
GAA P10253 2/20 0.35
TSHR P16473 1/20 0.35
TP53 P04637 1/20 0.35
POLB P06746 1/20 0.35
PTPN2 P17706 1/20 0.34
PTPN1 P18031 1/20 0.34
STAT3 P40763 1/20 0.34
PTPRS Q13332 1/20 0.34
PDK1 Q15118 1/20 0.34
PDK2 Q15119 1/20 0.34
PDK3 Q15120 1/20 0.34
PDK4 Q16654 1/20 0.34
MAPT P10636 2/20 0.34
NPSR1 Q6W5P4 1/20 0.34
PKLR P30613 2/20 0.34
HTT P42858 1/20 0.33
HTR7 P34969 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6984183 0.93 F2 (0.40) F2ALDH1A1GAATSHRTP53
SCHEMBL7958921 0.91 F2 (0.52) F2ALDH1A1GAATSHRTP53
SCHEMBL6978633 0.88 RORC (0.36) ALDH1A1TSHRTP53POLBPDK1
SCHEMBL7407618 0.88 ALDH1A1 (0.44) F2ALDH1A1GAATSHRPTPN2
SCHEMBL6979171 0.86 USP2 (0.41) ALDH1A1GAATSHRPOLBPDK1
SCHEMBL7089638 0.85 PARP1 (0.36) ALDH1A1GAATP53POLBPTPN2
SCHEMBL6984481 0.85 F2 (0.41) F2ALDH1A1GAATSHRTP53
SCHEMBL6976662 0.82 F2 (0.60) F2ALDH1A1GAAPOLBPTPN2
Hydrochloric Acid SCHEMBL6979622 0.81 F2 (0.39) F2ALDH1A1TSHRPOLBPDK1
SCHEMBL6984189 0.80 F2 (0.39) F2ALDH1A1GAATSHRTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed
US-6300342-B1 FOR THERAPY OR INHIBITING THROMBUS FORMATION; FOR THERAPY OF FIBRIN-DEPENDENT INFLAMMATORY CONDITION BOEHRINGER INGELHEIM PHARM KG (DE) 2001-10-09 US disclosed
EP-0991624-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT Boehringer Ingelheim Pharma KG (DE) 2000-04-12 EP disclosed
WO-1999000371-A1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA KG (DE) 1999-01-07 WO disclosed