SCHEMBL6984881

SCHEMBL6984881

O=C(c1cccc2cccnc12)N1CCOCC1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM4 Q14833 2/20 0.54
SMN1; SMN2 Q16637 5/20 0.53
ALDH1A1 P00352 2/20 0.53
PARP1 P09874 1/20 0.53
OPRM1 P35372 1/20 0.52
OPRD1 P41143 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
MEN1 O00255 1/20 0.52
KMT2A Q03164 1/20 0.52
HTT P42858 1/20 0.51
HCRTR1 O43613 1/20 0.51
HCRTR2 O43614 1/20 0.51
KDM4E B2RXH2 1/20 0.51
MAPT P10636 1/20 0.51
CCR3 P51677 1/20 0.50
GAA P10253 1/20 0.50
HTR2A P28223 1/20 0.50
HTR2C P28335 1/20 0.50
RIPK1 Q13546 1/20 0.49
NPSR1 Q6W5P4 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6986212 0.85 MAPT (0.59) SMN1; SMN2ALDH1A1PARP1OPRM1OPRD1
SCHEMBL2143749 0.85 ALDH1A1 (0.57) GRM4SMN1; SMN2ALDH1A1L3MBTL1HTT
SCHEMBL30073359 0.79 POLB (0.60) SMN1; SMN2ALDH1A1HTTKDM4EMAPT
SCHEMBL12844486 0.79 SMN1; SMN2 (0.55) SMN1; SMN2ALDH1A1HTTKDM4EMAPT
SCHEMBL855339 0.79 POLB (0.60) SMN1; SMN2ALDH1A1HTTKDM4EMAPT
SCHEMBL4159437 0.78 PARP1 (0.54) SMN1; SMN2ALDH1A1PARP1HTTHCRTR1
SCHEMBL19894106 0.78 HCRTR1 (0.60) HCRTR1HCRTR2CCR3HTR2AHTR2C
SCHEMBL27253846 0.78 KDM4E (0.58) GRM4SMN1; SMN2ALDH1A1L3MBTL1MEN1
SCHEMBL23775498 0.78 HTR2A (0.51) GRM4ALDH1A1PARP1OPRM1OPRD1
SCHEMBL16003034 0.78 HTR2A (0.53) GRM4PARP1HCRTR1HCRTR2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0991624-B1 PHENYLALKYL DERIVATIVES WITH THROMBIN-INHIBITING EFFECT BOEHRINGER INGELHEIM PHARMA (DE) 2003-11-19 EP disclosed