SCHEMBL6985293

SCHEMBL6985293

Nc1[c]cc2c(N)nc(-c3cc(N)c4ccnc(N)c4c3)cc2c1

nearest known ligand 0.32

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
SYK P43405 1/20 0.32
ACHE P22303 1/20 0.31
PDPK1 O15530 1/20 0.30
F12 P00748 1/20 0.30
PLAU P00749 1/20 0.30
NCF1 P14598 1/20 0.30
NOS3 P29474 1/20 0.30
NOS1 P29475 1/20 0.30
NOS2 P35228 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6161612 0.75 ROCK1 (0.47) F12PLAUNCF1NOS3NOS1
SCHEMBL18300458 0.60 ROCK1 (0.45) F12PLAUNCF1NOS3NOS1
SCHEMBL6162601 0.60 ROCK1 (0.45) F12PLAUNCF1NOS3NOS1
SCHEMBL6161145 0.60 ROCK1 (0.41) PDPK1F12PLAUNCF1NOS3
SCHEMBL6163883 0.59 NOS3 (0.41) F12PLAUNCF1NOS3NOS1
SCHEMBL24493428 0.55 MAP4K1 (0.38) F12PLAUNCF1NOS3NOS1
SCHEMBL509491 0.55 NPC1 (0.43) SYK
SCHEMBL14931471 0.55 ALDH1A1 (0.59) F12PLAUNCF1NOS3NOS1
SCHEMBL29508482 0.55 ALDH1A1 (0.59) F12PLAUNCF1NOS3NOS1
SCHEMBL509564 0.55 ADORA2A (0.47)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1175419-B1 ARYL SULFONYLS AS FACTOR XA INHIBITORS BRISTOL MYERS SQUIBB PHARMA CO (US) 2003-05-28 EP claimed