SCHEMBL6986308

SCHEMBL6986308

C=CCC(C)(C#N)c1ccc(Cl)c(Cl)c1

nearest known ligand 0.40

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
ESR1 P03372 1/20 0.35
ESR2 Q92731 1/20 0.35
AR P10275 2/20 0.35
KIF11 P52732 2/20 0.32
CASR P41180 1/20 0.31
MAPT P10636 1/20 0.30
SSTR4 P31391 1/20 0.30
SLC6A2 P23975 1/20 0.30
SLC6A4 P31645 1/20 0.30
SLC6A3 Q01959 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14390738 0.77 TSHR (0.40) TSHRESR1ESR2ARKIF11
SCHEMBL19237292 0.77 TSHR (0.40) TSHRESR1ESR2ARKIF11
SCHEMBL604108 0.77 TSHR (0.50) TSHRARKIF11CASRMAPT
SCHEMBL13946948 0.75 TSHR (0.41) TSHRKIF11CASRSSTR4SLC6A2
SCHEMBL28778794 0.74 TSHR (0.40) TSHRKIF11CASRSSTR4SLC6A2
SCHEMBL5779039 0.74 ALDH1A1 (0.46) TSHRESR1ESR2MAPT
SCHEMBL6990801 0.73 TSHR (0.39) TSHRKIF11CASRSLC6A2SLC6A4
SCHEMBL5879396 0.73 SIGMAR1 (0.36) TSHRKIF11
SCHEMBL13946950 0.72 TSHR (0.38) TSHRKIF11CASRSSTR4SLC6A2
SCHEMBL4026261 0.72 TSHR (0.41) TSHRKIF11SSTR4SLC6A2SLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1370520-A1 ARYL AND BIARYL COMPOUNDS HAVING MCH MODULATORY ACTIVITY PHARMACOPEIA, INC. (US) 2003-12-17 EP disclosed
WO-2002076929-A1 ARYL AND BIARYL COMPOUNDS HAVING MCH MODULATORY ACTIVITY PHARMACOPEIA, INC. (US) 2002-10-03 WO disclosed