SCHEMBL6986879

SCHEMBL6986879

COc1ccc(C(=O)c2cccc(NCC(=O)N3CCN(C4CCN(C)CC4)CC3)c2Cl)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 5/20 0.42
ALDH1A1 P00352 4/20 0.42
TSHR P16473 1/20 0.42
KDM4E B2RXH2 4/20 0.42
KDM1A O60341 3/20 0.42
MAOA P21397 2/20 0.42
MAOB P27338 2/20 0.42
ORAI1 Q96D31 1/20 0.42
ACHE P22303 2/20 0.41
PTGS2 P35354 1/20 0.41
TDP1 Q9NUW8 1/20 0.40
L3MBTL3 Q96JM7 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
F2 P00734 1/20 0.40
F10 P00742 1/20 0.40
HTR1F P30939 1/20 0.39
MAPT P10636 1/20 0.39
CHRM2 P08172 1/20 0.39
CHRM1 P11229 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6494015 0.99 KMT2A (0.41) KMT2AALDH1A1TSHRKDM4EKDM1A
SCHEMBL6986369 0.88 ALDH1A1 (0.41) KMT2AALDH1A1TSHRKDM4EKDM1A
Hydrochloric Acid SCHEMBL6986450 0.87 ALDH1A1 (0.40) KMT2AALDH1A1TSHRKDM4EKDM1A
SCHEMBL6986945 0.82 F10 (0.53) ALDH1A1KDM4EL3MBTL3L3MBTL1F2
Hydrochloric Acid SCHEMBL6985167 0.82 F10 (0.53) ALDH1A1KDM4EL3MBTL3L3MBTL1F2
Hydrochloric Acid SCHEMBL6980263 0.79 MAPT (0.46) KMT2AL3MBTL1MAPT
SCHEMBL6986644 0.78 F10 (0.43) KMT2AALDH1A1ACHEF10CHRM2
Hydrochloric Acid SCHEMBL6583478 0.77 F10 (0.46) KMT2AALDH1A1KDM4EACHEF10
SCHEMBL4832356 0.77 KRAS (0.51) ALDH1A1KDM4EKDM1AMAOBACHE
SCHEMBL6582418 0.76 SMO (0.40) KMT2AKDM4EF10MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289972-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP claimed
WO-2001096323-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO claimed
EP-1289972-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096323-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed