SCHEMBL6986369

SCHEMBL6986369

COc1ccc(C(=O)c2cccc(NCC(=O)N3CCN(C4CCN(C)CC4)CC3)c2C(F)(F)F)cc1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.41
KMT2A Q03164 2/20 0.41
TSHR P16473 1/20 0.41
SLC6A5 Q9Y345 4/20 0.41
KDM4E B2RXH2 2/20 0.41
ORAI1 Q96D31 1/20 0.41
ACHE P22303 2/20 0.40
PTGS2 P35354 1/20 0.40
TDP1 Q9NUW8 1/20 0.39
L3MBTL3 Q96JM7 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
KDM1A O60341 1/20 0.39
MAOA P21397 1/20 0.39
MAOB P27338 1/20 0.39
STAT3 P40763 1/20 0.38
CHRM2 P08172 2/20 0.38
CHRM1 P11229 2/20 0.38
MAPT P10636 1/20 0.38
SLC6A4 P31645 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6986450 0.99 ALDH1A1 (0.40) ALDH1A1KMT2ATSHRSLC6A5KDM4E
SCHEMBL6986879 0.88 KMT2A (0.42) ALDH1A1KMT2ATSHRKDM4EORAI1
Hydrochloric Acid SCHEMBL6494015 0.87 KMT2A (0.41) ALDH1A1KMT2ATSHRKDM4EORAI1
SCHEMBL6985018 0.84 F10 (0.49) ALDH1A1KDM4EL3MBTL3L3MBTL1STAT3
Hydrochloric Acid SCHEMBL6582680 0.78 F10 (0.45) ALDH1A1KMT2AKDM4EACHEMEN1
Hydrochloric Acid SCHEMBL6582721 0.78 F10 (0.40) ALDH1A1KMT2AKDM4EMEN1NPC1
SCHEMBL4832287 0.77 SCD (0.50) ALDH1A1TSHRKDM4EACHEL3MBTL3
SCHEMBL4844807 0.72 KDM4E (0.52) ALDH1A1KMT2AKDM4EACHEL3MBTL3
Hydrochloric Acid SCHEMBL6982358 0.72 ROCK2 (0.41) ALDH1A1KMT2AACHEMAPTHRH3
SCHEMBL4832356 0.71 KRAS (0.51) ALDH1A1KDM4EACHEL3MBTL3L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289972-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP claimed
WO-2001096323-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO claimed