SCHEMBL6987188

SCHEMBL6987188

CCc1cc2ccccc2n1-c1ccc(N)c(Cc2c(F)cccc2Cl)c1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
HTT P42858 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
NPC1 O15118 1/20 0.36
PPP1CA P62136 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
REN P00797 1/20 0.35
TAAR1 Q96RJ0 1/20 0.34
ALDH1A1 P00352 2/20 0.33
HPGD P15428 1/20 0.33
CYP19A1 P11511 1/20 0.33
MAPT P10636 3/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
DAO P14920 1/20 0.32
TP53 P04637 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6987190 0.77 ALDH1A1 (0.54) HTTSMN1; SMN2TDP1L3MBTL1ALDH1A1
SCHEMBL6985367 0.67 CYP19A1 (0.39) NPC1L3MBTL1ALDH1A1CYP19A1MAPT
SCHEMBL1878657 0.65 CYP19A1 (0.55) HTTL3MBTL1ALDH1A1HPGDCYP19A1
SCHEMBL11777239 0.64 MPO (0.44) HTTSMN1; SMN2TDP1TAAR1ALDH1A1
SCHEMBL9901553 0.63 ALDH1A1 (0.50) HTTSMN1; SMN2NPC1TDP1L3MBTL1
SCHEMBL22231717 0.63 TAAR1 (0.45) HTTSMN1; SMN2NPC1PPP1CATDP1
SCHEMBL6693208 0.63 TAAR1 (0.45) HTTSMN1; SMN2NPC1PPP1CATDP1
SCHEMBL31470103 0.62 HTT (0.51) HTTSMN1; SMN2NPC1PPP1CATDP1
SCHEMBL30023693 0.62 MPO (0.41) HTTSMN1; SMN2NPC1TDP1TAAR1
SCHEMBL805461 0.61 TAAR1 (0.61) HTTSMN1; SMN2TDP1TAAR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303508-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS Boehringer Ingelheim Pharmaceuticals, Inc. (US) 2003-04-23 EP disclosed
WO-2002006273-A1 SUBSTITUTED 1-(4-AMINOPHENYL)INDOLES AND THEIR USE AS ANTI-INFLAMMATORY AGENTS BOEHRINGER INGELHEIM PHARMACEUTICALS, INC. (US) 2002-01-24 WO disclosed