SCHEMBL6987892

SCHEMBL6987892

O=C(CNc1ccccc1)N1CCN(CCc2nccs2)CC1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
FAAH O00519 1/20 0.42
ALDH1A1 P00352 2/20 0.42
TSHR P16473 2/20 0.42
HRH1 P35367 1/20 0.42
PTGS2 P35354 1/20 0.41
KCNA5 P22460 1/20 0.41
CYP3A4 P08684 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
NPSR1 Q6W5P4 2/20 0.40
P2RX7 Q99572 1/20 0.39
KDM4E B2RXH2 1/20 0.39
HTT P42858 1/20 0.39
EGLN1 Q9GZT9 1/20 0.39
HTR7 P34969 1/20 0.39
SIGMAR1 Q99720 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4837366 0.99 FAAH (0.41) FAAHALDH1A1TSHRHRH1PTGS2
SCHEMBL4836758 0.81 TP53 (0.58) FAAHALDH1A1TSHRKDM4E
SCHEMBL4840912 0.79 P2RX7 (0.53) FAAHP2RX7
Hydrochloric Acid SCHEMBL4840698 0.78 P2RX7 (0.52) FAAHTSHRP2RX7
Hydrochloric Acid SCHEMBL4832771 0.78 P2RX7 (0.52) FAAHTSHRP2RX7
SCHEMBL4832913 0.78 P2RX7 (0.46) FAAHALDH1A1P2RX7KDM4EEGLN1
SCHEMBL4832750 0.76 FAAH (0.43) FAAHALDH1A1TSHRNPSR1KDM4E
SCHEMBL4832544 0.76 TP53 (0.43) FAAHALDH1A1TSHRNPSR1P2RX7
SCHEMBL4836752 0.76 KDM4E (0.54) FAAHALDH1A1P2RX7KDM4E
SCHEMBL13779963 0.75 KDM1A (0.57) ALDH1A1PTGS2KDM4EHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289972-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2003-03-12 EP disclosed
WO-2001096323-A1 SERINE PROTEASE INHIBITORS ELI LILLY AND COMPANY (US) 2001-12-20 WO disclosed