SCHEMBL6987908

SCHEMBL6987908

COC[C@@](N)(CC/C=C\CNCC=N)C(=O)O

nearest known ligand 0.33

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
MEN1 O00255 1/20 0.31
ALDH1A1 P00352 1/20 0.31
CYP1A2 P05177 1/20 0.31
THRB P10828 1/20 0.31
KMT2A Q03164 1/20 0.31
ARG1 P05089 1/20 0.31
ARG2 P78540 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989001 0.86 MEN1 (0.45) NOS1NOS2MEN1ALDH1A1CYP1A2
SCHEMBL6992300 0.86 MEN1 (0.45) NOS1NOS2MEN1ALDH1A1CYP1A2
SCHEMBL6988773 0.82 ODC1 (0.42) MEN1ALDH1A1CYP1A2THRBKMT2A
SCHEMBL6195060 0.81 NOS1 (0.33) NOS1NOS2ARG1ARG2
SCHEMBL7075158 0.80 NOS1 (0.33) NOS1NOS2
SCHEMBL7071571 0.80 NOS1 (0.33) NOS1NOS2
Hydrochloric Acid SCHEMBL6192268 0.80 NOS1 (0.35) NOS1NOS2ARG1ARG2
SCHEMBL6992519 0.80 NOS1 (0.31) NOS1NOS2
SCHEMBL6994163 0.80 NOS1 (0.31) NOS1NOS2
SCHEMBL6992523 0.80 NOS1 (0.31) NOS1NOS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1317421-A1 2-AMINO-2-ALKYL-5 HEPTENOIC AND HEPTYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS Pharmacia Corporation (US) 2003-06-11 EP claimed
WO-2002022562-A1 2-AMINO-2-ALKYL-5 HEPTENOIC AND HEPTYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS PHARMACIA CORPORATION (US) 2002-03-21 WO claimed
EP-1317421-A1 2-AMINO-2-ALKYL-5 HEPTENOIC AND HEPTYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS Pharmacia Corporation (US) 2003-06-11 EP disclosed
WO-2002022562-A1 2-AMINO-2-ALKYL-5 HEPTENOIC AND HEPTYNOIC ACID DERIVATIVES USEFUL AS NITRIC OXIDE SYNTHASE INHIBITORS PHARMACIA CORPORATION (US) 2002-03-21 WO disclosed