SCHEMBL6989198

SCHEMBL6989198

C[C@H](N)CCCS(=O)(=O)Cc1cnc2ccccc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 2/20 0.43
PDE10A Q9Y233 5/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA9 Q16790 1/20 0.38
HIF1A Q16665 1/20 0.38
EPAS1 Q99814 1/20 0.38
MMP9 P14780 2/20 0.37
MMP1 P03956 1/20 0.37
FCER2 P06734 1/20 0.37
MMP3 P08254 1/20 0.37
KMT2A Q03164 2/20 0.37
RAB9A P51151 1/20 0.37
ALDH1A1 P00352 1/20 0.36
LMNA P02545 1/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
HTT P42858 1/20 0.36
MEN1 O00255 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL6985055 0.99 CYP1A2 (0.42) CYP1A2PDE10ACA12CA1CA2
SCHEMBL6988727 0.85 CYP1A2 (0.41) CYP1A2HIF1AEPAS1MMP9MMP1
SCHEMBL6988734 0.85 CYP1A2 (0.41) CYP1A2HIF1AEPAS1MMP9MMP1
SCHEMBL27578438 0.82 TRPV1 (0.44) CYP1A2PDE10AHIF1AEPAS1KMT2A
SCHEMBL6987672 0.82 HDAC3 (0.38) CYP1A2HIF1AEPAS1MMP9MMP1
SCHEMBL6987677 0.82 HDAC3 (0.38) CYP1A2HIF1AEPAS1MMP9MMP1
SCHEMBL6987203 0.81 CYP1A2 (0.38) CYP1A2PDE10AHIF1AEPAS1MMP9
SCHEMBL6988573 0.80 CYP1A2 (0.42) CYP1A2HIF1AEPAS1MMP9MMP1
SCHEMBL6989193 0.78 CYP1A2 (0.43) CYP1A2PDE10ACA12CA1CA2
SCHEMBL6982449 0.77 HIF1A (0.35) CYP1A2PDE10AHIF1AEPAS1MMP9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1289980-A1 BICYCLYL OR HETEROBICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED N-HYDROXYFORMAMIDES SMITHKLINE BEECHAM PLC (GB) 2003-03-12 EP disclosed
WO-2001090100-A1 BICYCLYL OR HETEROBICYCLYLMETHANESULFONYLAMINO-SUBSTITUTED N-HYDROXYFORMAMIDES SMITHKLINE BEECHAM P.L.C. (GB) 2001-11-29 WO disclosed