SCHEMBL6989320

SCHEMBL6989320

FC(F)(F)c1[c]ccc(-c2cccc(C(F)(F)F)c2)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.46
MAOB P27338 1/20 0.44
NOTUM Q6P988 2/20 0.42
KIF11 P52732 1/20 0.42
IDO1 P14902 1/20 0.41
TSHR P16473 1/20 0.41
MAPK1 P28482 1/20 0.41
PGR P06401 1/20 0.41
ASIC3 Q9UHC3 1/20 0.41
SCN2A Q99250 2/20 0.41
HTR2C P28335 2/20 0.40
CTSS P25774 1/20 0.40
CA12 O43570 1/20 0.39
CA9 Q16790 1/20 0.39
PARP1 P09874 1/20 0.39
ALDH1A1 P00352 1/20 0.38
GAA P10253 1/20 0.38
ATM Q13315 1/20 0.38
PARP10 Q53GL7 1/20 0.38
PARP11 Q9NR21 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1068350 0.83 KIF11 (0.43) KDM1AKIF11TSHRALDH1A1
SCHEMBL145774 0.82 MAOB (0.44) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL2430768 0.82 NT5E (0.43) NOTUMIDO1CA12CA9
SCHEMBL5198912 0.81 ALOX5 (0.41) MAOBNOTUMIDO1TSHRPGR
SCHEMBL143472 0.81 IKBKB (0.43) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL695494 0.81 MAOB (0.43) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL29678302 0.80 TSHR (0.58) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL1263144 0.80 TSHR (0.58) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL142774 0.79 MAOB (0.51) KDM1AMAOBNOTUMKIF11IDO1
SCHEMBL6988230 0.79 KDM1A (0.50) KDM1AMAOBNOTUMKIF11IDO1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1318985-A2 4-AMINO-QUINAZOLINES MERCK PATENT GmbH (DE) 2003-06-18 EP disclosed
WO-2002024666-A2 4-AMINO-QUINAZOLINES MERCK PATENT GMBH (DE) 2002-03-28 WO disclosed