SCHEMBL6989536

SCHEMBL6989536

COc1cc2c(cc1OC)[C@H]([C@H]1CCC(=O)O1)N(C(=O)OCc1ccccc1)CC2

nearest known ligand 0.75

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 8/20 0.49
ALDH1A1 P00352 3/20 0.47
MAPT P10636 2/20 0.47
HPGD P15428 1/20 0.47
TSHR P16473 1/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
TRPV1 Q8NER1 1/20 0.47
MTNR1A P48039 1/20 0.46
NPC1 O15118 1/20 0.46
MITF O75030 1/20 0.46
LMNA P02545 1/20 0.46
XBP1 P17861 1/20 0.46
HTT P42858 1/20 0.46
RAB9A P51151 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
KDM4E B2RXH2 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6989538 1.00 MTNR1B (0.49) MTNR1BALDH1A1MAPTHPGDTSHR
SCHEMBL7566815 0.86 PARP1 (0.48) SMN1; SMN2NPC1RAB9ANPSR1L3MBTL1
SCHEMBL6991074 0.86 PARP1 (0.48) SMN1; SMN2NPC1RAB9ANPSR1L3MBTL1
SCHEMBL6991071 0.86 PARP1 (0.48) SMN1; SMN2NPC1RAB9ANPSR1L3MBTL1
SCHEMBL29380426 0.86 PARP1 (0.48) SMN1; SMN2NPC1RAB9ANPSR1L3MBTL1
SCHEMBL7566816 0.86 PARP1 (0.48) SMN1; SMN2NPC1RAB9ANPSR1L3MBTL1
SCHEMBL7241406 0.83 MTNR1B (0.48) MTNR1BALDH1A1MAPTHPGDTSHR
SCHEMBL7241403 0.83 MTNR1B (0.48) MTNR1BALDH1A1MAPTHPGDTSHR
SCHEMBL5463056 0.79 TRPV1 (0.72) MTNR1BALDH1A1MAPTHPGDTSHR
SCHEMBL5464723 0.79 MTNR1B (0.61) MTNR1BTRPV1MTNR1ALMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649626-B1 Stimulants of gamma -aminobutyric acid receptors; psychological disorders CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2003-11-18 US disclosed
EP-1224182-B1 N-SUBSTITUTED 1-(BUTYROLACTONE)-ISOQUINOLINES FOR TREATING NERVOUS DISORDERS CENTRE NAT RECH SCIENT (FR) 2003-07-16 EP disclosed