SCHEMBL6991071

SCHEMBL6991071

O=C1CC[C@H]([C@H]2c3ccccc3CCN2C(=O)OCc2ccccc2)O1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 1/20 0.48
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
F2 P00734 2/20 0.46
ELANE P08246 2/20 0.46
CTSG P08311 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.42
NPSR1 Q6W5P4 1/20 0.42
PREP P48147 1/20 0.41
TMEM97 Q5BJF2 2/20 0.41
SIGMAR1 Q99720 2/20 0.41
CHRM4 P08173 1/20 0.41
HTR1A P08908 1/20 0.41
CHRM5 P08912 1/20 0.41
ADRA2A P08913 1/20 0.41
ADRA2B P18089 1/20 0.41
HRH2 P25021 1/20 0.41
ADRA1D P25100 1/20 0.41
HTR2A P28223 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6991074 1.00 PARP1 (0.48) PARP1NPC1RAB9AL3MBTL1F2
SCHEMBL29380426 1.00 PARP1 (0.48) PARP1NPC1RAB9AL3MBTL1F2
SCHEMBL7566815 1.00 PARP1 (0.48) PARP1NPC1RAB9AL3MBTL1F2
SCHEMBL7566816 1.00 PARP1 (0.48) PARP1NPC1RAB9AL3MBTL1F2
SCHEMBL6989536 0.86 MTNR1B (0.49) NPC1RAB9AL3MBTL1SMN1; SMN2NPSR1
SCHEMBL6989538 0.86 MTNR1B (0.49) NPC1RAB9AL3MBTL1SMN1; SMN2NPSR1
SCHEMBL6986196 0.76 P2RX4 (0.40) NPC1RAB9AL3MBTL1F2ELANE
SCHEMBL6986189 0.76 P2RX4 (0.40) NPC1RAB9AL3MBTL1F2ELANE
SCHEMBL1052868 0.76 ACE (0.58) PARP1NPC1RAB9AL3MBTL1SMN1; SMN2
SCHEMBL14646661 0.76 NPC1 (0.55) PARP1NPC1RAB9AL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6649626-B1 Stimulants of gamma -aminobutyric acid receptors; psychological disorders CENTRE NATIONAL DE LA RECHERCHE SCIENTIFIQUE (CNRS) (FR) 2003-11-18 US disclosed
EP-1224182-B1 N-SUBSTITUTED 1-(BUTYROLACTONE)-ISOQUINOLINES FOR TREATING NERVOUS DISORDERS CENTRE NAT RECH SCIENT (FR) 2003-07-16 EP disclosed