SCHEMBL6990370

SCHEMBL6990370

CS(=O)(=O)c1cc(N2CCCC(F)(NS(=O)(=O)c3cnc(Cl)c(Br)c3)C2=O)ccc1-c1ccccc1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 11/20 0.36
GAA P10253 1/20 0.36
MAPT P10636 1/20 0.36
JAK2 O60674 1/20 0.36
PKM P14618 1/20 0.36
MCOLN3 Q8TDD5 1/20 0.36
LMNA P02545 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
F10 P00742 2/20 0.35
HTT P42858 3/20 0.35
DRD2 P14416 1/20 0.34
ADRA1D P25100 1/20 0.34
ADRA1A P35348 1/20 0.34
ADRA1B P35368 1/20 0.34
EIF2AK3 Q9NZJ5 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4680196 0.92 F10 (0.41) ALDH1A1GAAMAPTJAK2PKM
SCHEMBL6989555 0.85 F10 (0.43) ALDH1A1GAAMAPTLMNAL3MBTL1
SCHEMBL6985447 0.84 F10 (0.45) F10DRD2
SCHEMBL6980681 0.84 F10 (0.45) ALDH1A1MAPTLMNANPSR1F10
SCHEMBL6986546 0.83 F10 (0.42) F10HTT
SCHEMBL6985663 0.81 F10 (0.45) LMNAF10DRD2
SCHEMBL6988024 0.81 F10 (0.45) ALDH1A1GAAMAPTLMNAL3MBTL1
SCHEMBL6985337 0.79 LMNA (0.40) ALDH1A1GAAPKMLMNAF10
SCHEMBL6992512 0.79 F10 (0.46) L3MBTL1F10
SCHEMBL6982192 0.79 F10 (0.38) F10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1337251-A1 MONOCYCLIC OR BICYCLIC CARBOCYCLES AND HETEROCYCLES AS FACTOR XA INHIBITORS Bristol-Myers Squibb Pharma Company (US) 2003-08-27 EP claimed
WO-2002102380-A1 MONOCYCLIC OR BICYCLIC CARBOCYCLES AND HETEROCYCLES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-12-27 WO claimed
EP-1337251-A1 MONOCYCLIC OR BICYCLIC CARBOCYCLES AND HETEROCYCLES AS FACTOR XA INHIBITORS Bristol-Myers Squibb Pharma Company (US) 2003-08-27 EP disclosed
WO-2002102380-A1 MONOCYCLIC OR BICYCLIC CARBOCYCLES AND HETEROCYCLES AS FACTOR XA INHIBITORS BRISTOL-MYERS SQUIBB PHARMA COMPANY (US) 2002-12-27 WO disclosed