SCHEMBL6991657

SCHEMBL6991657

COc1ccc2[nH]c(=O)c(-c3ccccc3)c(OC(=O)O)c2c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.53
HPGD P15428 4/20 0.53
PADI4 Q9UM07 2/20 0.52
TUBB4A P04350 1/20 0.50
TUBB P07437 1/20 0.50
TUBA3C P0DPH7 1/20 0.50
TUBA1B P68363 1/20 0.50
TUBA4A P68366 1/20 0.50
TUBB4B P68371 1/20 0.50
TUBB3 Q13509 1/20 0.50
TUBB2A Q13885 1/20 0.50
TUBB8 Q3ZCM7 1/20 0.50
TUBA3E Q6PEY2 1/20 0.50
TUBA1A Q71U36 1/20 0.50
TUBA1C Q9BQE3 1/20 0.50
TUBB6 Q9BUF5 1/20 0.50
TUBB2B Q9BVA1 1/20 0.50
TUBB1 Q9H4B7 1/20 0.50
MAPK10 P53779 1/20 0.48
MTNR1A P48039 3/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7002128 0.87 ALDH1A1 (0.47) ALDH1A1HPGDPADI4TUBB4ATUBB
SCHEMBL8182316 0.82 PADI4 (0.56) ALDH1A1HPGDPADI4TUBB4ATUBB
SCHEMBL6998713 0.82 MAPT (0.60) ALDH1A1HPGDPADI4KDM4EGAA
SCHEMBL8189447 0.77 PADI4 (0.51) ALDH1A1HPGDPADI4TUBB4ATUBB
SCHEMBL4827488 0.74 CYP1A2 (0.62) ALDH1A1HPGDKDM4EPOLBHSD17B10
SCHEMBL6995868 0.74 KDM4E (0.64) ALDH1A1HPGDGSK3AGSK3BKDM4E
SCHEMBL10648743 0.73 MAPT (0.59) ALDH1A1HPGDPADI4TUBB4ATUBB
SCHEMBL7825662 0.72 PADI4 (0.57) ALDH1A1HPGDPADI4TUBB4ATUBB
SCHEMBL18019742 0.72 ALDH1A1 (0.57) ALDH1A1HPGDTUBB4ATUBBTUBA3C
SCHEMBL15060149 0.72 ALDH1A1 (0.61) ALDH1A1HPGDTUBB4ATUBBTUBA3C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1003724-B1 SUBSTITUTED QUINOLINE DERIVATIVES WITH ANTIVIRAL ACTION AVENTIS PHARMA GMBH (DE) 2003-02-12 EP disclosed
EP-1003724-A1 SUBSTITUTED QUINOLINE DERIVATIVES WITH ANTIVIRAL ACTION Aventis Pharma Deutschland GmbH (DE) 2000-05-31 EP disclosed
WO-1997037977-A1 SUBSTITUTED QUINOLINE DERIVATIVES WITH ANTIVIRAL ACTION HOECHST AKTIENGESELLSCHAFT (DE) 1997-10-16 WO disclosed