SCHEMBL6991660

SCHEMBL6991660

COc1cccc(C2=NC(=O)C(C)(C)O2)c1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 4/20 0.50
PGR P06401 3/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
NOTUM Q6P988 2/20 0.46
NCOA1 Q15788 1/20 0.45
NCOA3 Q9Y6Q9 1/20 0.45
DAPK3 O43293 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
DYRK1A Q13627 1/20 0.44
CLK4 Q9HAZ1 1/20 0.44
TDO2 P48775 1/20 0.43
GAA P10253 1/20 0.43
ALDH1A1 P00352 3/20 0.42
KMT2A Q03164 2/20 0.42
F2 P00734 1/20 0.42
KDM4E B2RXH2 2/20 0.42
USP2 O75604 1/20 0.42
CYP3A4 P08684 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6997691 0.73 NPC1 (0.40) HPGDPGRNPC1RAB9ANOTUM
SCHEMBL8383654 0.72 NISCH (0.46) HPGDPGRNPC1RAB9ANOTUM
SCHEMBL3041896 0.72 HPGD (0.51) HPGDNPC1RAB9ANOTUMNCOA1
SCHEMBL24534483 0.72 HPGD (0.61) HPGDNPC1RAB9ANOTUMNCOA1
SCHEMBL28613547 0.71 HDAC4 (0.51) HPGDPGRNOTUMNCOA1NCOA3
SCHEMBL24534874 0.70 NPC1 (0.74) HPGDNPC1RAB9ANOTUMDAPK3
SCHEMBL4158013 0.70 PGR (0.81) PGRNOTUMNCOA1NCOA3HDAC4
SCHEMBL29489425 0.69 CYP3A4 (0.73) NOTUMHDAC4HDAC8DYRK1ACLK4
SCHEMBL196765 0.69 CYP3A4 (0.73) NOTUMHDAC4HDAC8DYRK1ACLK4
SCHEMBL1996001 0.69 KDM4E (0.51) NOTUMNCOA1NCOA3DYRK1ACLK4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0863906-B1 HETEROCYCLIC DIOXETHANE SUBSTRATES, PROCESS FOR THEIR PREPARATION AND THEIR USE ROCHE DIAGNOSTICS GMBH (DE) 2003-02-12 EP disclosed
US-6107036-A Heterocyclic dioxethane substrates, process for their preparation and their use ROCHE DIAGNOSTICS GMBH (DE) 2000-08-22 US disclosed
EP-0863906-A2 HETEROCYCLIC DIOXETHANE SUBSTRATES, PROCESS FOR THEIR PREPARATION AND THEIR USE Roche Diagnostics GmbH (DE) 1998-09-16 EP disclosed
WO-1997014696-A2 HETEROCYCLIC DIOXETHANE SUBSTRATES, PROCESS FOR THEIR PREPARATION AND THEIR USE BOEHRINGER MANNHEIM GMBH (DE) 1997-04-24 WO disclosed