SCHEMBL6992191

SCHEMBL6992191

COc1ccccc1N1CCN(CCCN2CCC(=NO)c3ccn(C)c3C2=O)CC1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 14/20 0.62
DRD2 P14416 13/20 0.59
DRD4 P21917 8/20 0.59
DRD1 P21728 3/20 0.58
HTR7 P34969 2/20 0.53
DRD5 P21918 1/20 0.53
ALDH1A1 P00352 2/20 0.52
MEN1 O00255 1/20 0.52
CYP3A4 P08684 1/20 0.52
HTR1A P08908 1/20 0.52
CYP2D6 P10635 1/20 0.52
ALOX12 P18054 1/20 0.52
ADRA1D P25100 1/20 0.52
ADRA1A P35348 1/20 0.52
ADRA1B P35368 1/20 0.52
KMT2A Q03164 1/20 0.52
HIF1A Q16665 1/20 0.52
HSD17B10 Q99714 1/20 0.52
KDM4E B2RXH2 1/20 0.52
GLA P06280 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6992184 1.00 DRD3 (0.62) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6990417 0.88 DRD3 (0.67) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6992608 0.85 HTR1A (0.48) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6992602 0.85 HTR1A (0.48) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6994634 0.84 DRD3 (0.59) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6994638 0.84 DRD3 (0.59) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6993732 0.83 DRD2 (0.59) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6993734 0.83 DRD2 (0.59) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6989075 0.83 HTR1A (0.49) DRD3DRD2DRD4DRD1HTR7
SCHEMBL6989077 0.83 HTR1A (0.49) DRD3DRD2DRD4DRD1HTR7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0557526-B1 PYRROLOAZEPINE COMPOUND SUNTORY LTD (JP) 2003-04-02 EP disclosed
US-5399557-A Cardiovascular disorders SUNTORY LIMITED (JP) 1995-03-21 US disclosed
EP-0557526-A1 PYRROLOAZEPINE COMPOUND SUNTORY LIMITED (JP) 1993-09-01 EP disclosed