SCHEMBL6992595

SCHEMBL6992595

COc1ccc(-c2ccc3c(Cl)cnc(Cl)c3c2)cc1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PLAU P00749 5/20 0.65
PLG P00747 3/20 0.65
MAP4K4 O95819 1/20 0.46
DYRK1A Q13627 3/20 0.45
PLAT P00750 2/20 0.45
ABL1 P00519 1/20 0.40
ABCB1 P08183 1/20 0.40
BCR P11274 1/20 0.40
PDGFRB P09619 1/20 0.40
PDGFRA P16234 1/20 0.40
NPC1 O15118 3/20 0.40
RAB9A P51151 3/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
CASP3 P42574 1/20 0.40
SENP7 Q9BQF6 1/20 0.40
ALDH1A1 P00352 1/20 0.40
LMNA P02545 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6994679 0.89 PLAU (0.53) PLAUPLGMAP4K4PLATABL1
SCHEMBL1536456 0.87 PLAU (0.49) PLAUPLGDYRK1AKMT2AALDH1A1
SCHEMBL7001317 0.87 PLAU (0.67) PLAUPLGMAP4K4DYRK1APDGFRB
SCHEMBL6991093 0.85 PLAU (0.49) PLAUPLGMAP4K4DYRK1AABL1
SCHEMBL6998335 0.82 PLAU (0.62) PLAUPLGPLATNPC1RAB9A
SCHEMBL1536440 0.80 PLAU (0.46) PLAUPLGDYRK1AKMT2AALDH1A1
SCHEMBL6437504 0.79 PLAU (1.00) PLAUPLGPLAT
SCHEMBL6997008 0.78 PLAU (0.50) PLAUPLGPLATALDH1A1
SCHEMBL6437497 0.77 PLAU (0.63) PLAUPLGMAP4K4DYRK1APLAT
SCHEMBL6997835 0.77 PLAU (0.68) PLAUPLGMAP4K4PLATPDGFRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023268-B1 ISOQUINOLINES AS UROKINASE INHIBITORS PFIZER LTD (GB) 2003-05-21 EP disclosed
US-6248738-B1 ANTIULCER AGENTS, ANGIOGENESIS INHIBITORS, ANTIMETASTASIS AGENTS, ANTITUMOR AGENTS PFIZER INC. 2001-06-19 US disclosed