SCHEMBL6993535

SCHEMBL6993535

Cc1ccc(-c2ccccc2C(=O)Nc2ccc(C(=O)N3CCc4nc(C)oc4-c4ccccc43)cc2)cc1

nearest known ligand 0.59

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
AVPR2 P30518 12/20 0.59
AVPR1A P37288 8/20 0.59
OXTR P30559 1/20 0.53
AVPR1B P47901 4/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6619403 0.95 AVPR2 (0.65) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL6987926 0.83 AVPR2 (0.68) AVPR2AVPR1AOXTRAVPR1B
Hydrochloric Acid SCHEMBL6988764 0.82 AVPR2 (0.67) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL8961694 0.81 AVPR2 (0.72) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL1495876 0.80 ALDH1A1 (0.49) AVPR2AVPR1A
SCHEMBL6989484 0.80 AVPR2 (0.70) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL6994936 0.80 AVPR2 (0.62) AVPR2AVPR1AOXTRAVPR1B
SCHEMBL6972323 0.78 AVPR2 (0.80) AVPR2AVPR1AOXTR
SCHEMBL6955045 0.78 AVPR2 (0.85) AVPR2AVPR1AOXTRAVPR1B
Conivaptan SCHEMBL29406590 0.78 AVPR2 (0.75) AVPR2AVPR1AOXTRAVPR1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0709386-B1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMA CO LTD (JP) 2003-05-07 EP disclosed
EP-1097920-A1 Intermediate for condensed benzazepine derivatives YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 2001-05-09 EP disclosed
EP-0709386-A1 FUSED BENZAZEPINE DERIVATIVE AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1996-05-01 EP disclosed