SCHEMBL6994817

SCHEMBL6994817

O=CC(c1ccccc1)N1CC(F)(F)Cn2c1nc(-c1ccncn1)cc2=O

nearest known ligand 0.42

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 20/20 0.42
CYP2D6 P10635 6/20 0.41
CYP1A2 P05177 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3565547 0.75 GSK3B (0.45) GSK3BCYP2D6CYP1A2
SCHEMBL6225885 0.74 GSK3B (0.53) GSK3BCYP2D6CYP1A2
SCHEMBL6995827 0.72 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL3566871 0.71 GSK3B (0.49) GSK3BCYP2D6CYP1A2
SCHEMBL3568873 0.71 GSK3B (0.46) GSK3BCYP2D6CYP1A2
SCHEMBL3568800 0.70 GSK3B (0.41) GSK3BCYP2D6CYP1A2
SCHEMBL3367409 0.69 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3370809 0.69 GSK3B (0.47) GSK3BCYP2D6CYP1A2
SCHEMBL3568346 0.69 GSK3B (0.43) GSK3BCYP2D6CYP1A2
SCHEMBL4576867 0.69 GSK3B (0.40) GSK3BCYP2D6CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1340760-A1 Substituted 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-one and 7-pyrimidinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5(1H)one derivatives SANOFI-SYNTHELABO (FR) 2003-09-03 EP disclosed
EP-1295884-A1 2-pyrimidinyl-6,7,8,9-tetrahydropyrimido[1,2-a]Pyrimidin-4-one and 7-Pyrimidinyl-2,3-Dihydroimidazo[1,2-a]Pyrimidin-5(1H)one derivatives SANOFI-SYNTHELABO (FR) 2003-03-26 EP disclosed