SCHEMBL6995124

SCHEMBL6995124

COc1ccc(CCC(C)(C)OC(=O)C(N)c2ccc3c(c2)NC(=O)C(C)O3)cc1

nearest known ligand 0.41

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 7/20 0.41
HTR1A P08908 2/20 0.40
HTR7 P34969 2/20 0.40
KCNH2 Q12809 1/20 0.38
HSD17B10 Q99714 3/20 0.38
SMYD3 Q9H7B4 3/20 0.35
DAO P14920 1/20 0.34
KDM4E B2RXH2 1/20 0.33
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000925 0.91 PARP1 (0.42) PARP1SMYD3POLB
SCHEMBL6998537 0.91 PARP1 (0.41) PARP1HTR1AHTR7KCNH2HSD17B10
SCHEMBL6999457 0.90 PARP1 (0.42) PARP1HSD17B10SMYD3ALDH1A1POLB
SCHEMBL6991397 0.89 PARP1 (0.40) PARP1HTR1AHTR7HSD17B10SMYD3
SCHEMBL7003521 0.88 PARP1 (0.39) PARP1HTR1AHTR7SMYD3MAPK1
SCHEMBL7001819 0.87 PARP1 (0.39) PARP1SMYD3KDM4EALDH1A1POLB
SCHEMBL7001012 0.87 PARP1 (0.40) PARP1SMYD3ALDH1A1POLB
SCHEMBL6996225 0.86 PARP1 (0.39) PARP1SMYD3ALDH1A1POLB
SCHEMBL7000920 0.85 PARP1 (0.41) PARP1HTR1AHTR7SMYD3DAO
SCHEMBL6994403 0.85 PARP1 (0.41) PARP1HSD17B10SMYD3DAOALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed