SCHEMBL7001819

SCHEMBL7001819

CC1Oc2ccc(C(N)C(=O)OC(C)(C)CCc3ccc([N+](=O)[O-])cc3)cc2NC1=O

nearest known ligand 0.39

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 8/20 0.39
SMYD3 Q9H7B4 3/20 0.34
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
PDE3B Q13370 1/20 0.32
PDE3A Q14432 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM4E B2RXH2 1/20 0.32
USP2 O75604 1/20 0.32
LMNA P02545 1/20 0.32
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7000745 0.91 PARP1 (0.39) PARP1SMYD3POLBPDE3AKMT2A
SCHEMBL7000925 0.89 PARP1 (0.42) PARP1SMYD3POLBUSP2
SCHEMBL6996238 0.88 PARP1 (0.41) PARP1SMYD3PDE3BPDE3AUSP2
SCHEMBL6999457 0.88 PARP1 (0.42) PARP1SMYD3ALDH1A1POLBLMNA
SCHEMBL7003826 0.88 PARP1 (0.39) PARP1SMYD3PDE3BPDE3AKMT2A
SCHEMBL7003521 0.88 PARP1 (0.39) PARP1SMYD3PDE3BPDE3A
SCHEMBL6995124 0.87 PARP1 (0.41) PARP1SMYD3ALDH1A1POLBKDM4E
SCHEMBL6991397 0.87 PARP1 (0.40) PARP1SMYD3PDE3BPDE3AKDM4E
SCHEMBL7001012 0.85 PARP1 (0.40) PARP1SMYD3ALDH1A1POLBPDE3B
SCHEMBL6996225 0.84 PARP1 (0.39) PARP1SMYD3ALDH1A1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-B1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AG (DE) 2003-12-03 EP disclosed