SCHEMBL6995202

SCHEMBL6995202

N#Cc1ccc2ccn(CC3CCN(CCc4ccc(F)cc4)C3)c2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HRH3 Q9Y5N1 2/20 0.45
HTR2A P28223 4/20 0.42
CCR3 P51677 2/20 0.42
KCNJ1 P48048 1/20 0.41
KCNH2 Q12809 1/20 0.41
KDM4E B2RXH2 2/20 0.40
ALDH1A1 P00352 2/20 0.40
TSHR P16473 2/20 0.40
HSD17B10 Q99714 2/20 0.40
USP2 O75604 1/20 0.40
POLB P06746 1/20 0.40
HPGD P15428 1/20 0.40
DRD2 P14416 3/20 0.39
DRD3 P35462 1/20 0.39
HTR2C P28335 3/20 0.39
HTR7 P34969 1/20 0.39
HTR6 P50406 1/20 0.39
HTR2B P41595 2/20 0.39
SIGMAR1 Q99720 2/20 0.39
MAOA P21397 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL7953973 0.99 HRH3 (0.44) HRH3HTR2ACCR3KCNJ1KCNH2
SCHEMBL7002079 0.90 DRD2 (0.50) HRH3CCR3KCNJ1KCNH2KDM4E
SCHEMBL6998697 0.89 HRH3 (0.43) HRH3HTR2ACCR3KCNH2KDM4E
Hydrochloric Acid SCHEMBL7952278 0.89 DRD2 (0.49) HRH3CCR3KCNJ1KCNH2KDM4E
Hydrochloric Acid SCHEMBL7954300 0.89 HRH3 (0.42) HRH3HTR2ACCR3KCNH2KDM4E
SCHEMBL6998142 0.87 HRH3 (0.45) HRH3SIGMAR1MAOB
SCHEMBL6991629 0.87 HRH3 (0.51) HRH3KDM4EALDH1A1TSHRHSD17B10
Hydrochloric Acid SCHEMBL7943915 0.87 HRH3 (0.44) HRH3KCNH2SIGMAR1MAOB
Hydrochloric Acid SCHEMBL7943799 0.86 HRH3 (0.50) HRH3KDM4EALDH1A1TSHRHSD17B10
SCHEMBL7000086 0.84 DRD2 (0.52) HTR2ACCR3KDM4EALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1023898-B1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands SERVIER LAB (FR) 2003-03-12 EP disclosed
EP-1023898-A1 Cyano-indoles as serotonine reuptake inhibitors and as 5-HT2c receptor ligands ADIR ET COMPAGNIE (FR) 2000-08-02 EP disclosed