SCHEMBL6995330

SCHEMBL6995330

CC(C)(C)NS(=O)(=O)c1ccccc1-c1ccc(NC(=O)O)cc1.N=C(NO)c1cccc(NC2CCCCC2)c1

nearest known ligand 0.42

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
F10 P00742 10/20 0.42
FPR2 P25090 2/20 0.41
FPR1 P21462 1/20 0.41
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
USP30 Q70CQ3 3/20 0.39
GPR119 Q8TDV5 1/20 0.38
IDO1 P14902 1/20 0.38
LMNA P02545 1/20 0.38
PRSS1 P07477 4/20 0.37
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
F2 P00734 1/20 0.36
KCNH2 Q12809 1/20 0.36
PRSS2 P07478 2/20 0.36
PRSS3 P35030 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6993750 0.99 FPR2 (0.42) F10FPR2FPR1CYP3A4CYP2D6
SCHEMBL6999615 0.91 F10 (0.52) F10PRSS1F2KCNH2PRSS2
SCHEMBL6993192 0.90 F10 (0.44) F10FPR2IDO1PRSS1F2
SCHEMBL6989579 0.89 PRSS1 (0.44) F10FPR2IDO1PRSS1F2
SCHEMBL6991785 0.88 F10 (0.54) F10PRSS1F2KCNH2PRSS2
SCHEMBL6996683 0.88 F10 (0.53) F10PRSS1F2KCNH2PRSS2
SCHEMBL7093219 0.84 USP30 (0.45) F10FPR2FPR1CYP3A4CYP2D6
SCHEMBL7143506 0.83 USP30 (0.44) F10FPR2FPR1CYP3A4CYP2D6
SCHEMBL7401213 0.81 F10 (0.40) F10PRSS1F2KCNH2PRSS2
SCHEMBL6988107 0.81 F10 (0.55) F10PRSS1F2KCNH2PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1303482-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GmbH (DE) 2003-04-23 EP disclosed
WO-2002008177-A2 N-SUBSTITUTED-1-AMINO-1,1-DIALKYLCARBOXYLIC ACID DERIVATIVES MERCK PATENT GMBH (DE) 2002-01-31 WO disclosed