SCHEMBL6995574

SCHEMBL6995574

COCCc1ccc(C)cc1N

nearest known ligand 0.47

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.47
CYP3A4 P08684 2/20 0.47
TDP1 Q9NUW8 2/20 0.45
ALOX15 P16050 2/20 0.45
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 1/20 0.42
HSD17B10 Q99714 1/20 0.41
SLC6A4 P31645 6/20 0.40
SLC6A2 P23975 4/20 0.40
SLC6A3 Q01959 4/20 0.40
CA1 P00915 1/20 0.39
TAAR1 Q96RJ0 1/20 0.37
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5252467 0.83 TDP1 (0.56) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL2131106 0.82 GAA (0.46) ALDH1A1CYP3A4TDP1TP53KDM4E
SCHEMBL18579434 0.80 ALDH1A1 (0.50) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL3580131 0.79 ALDH1A1 (0.48) ALDH1A1CYP3A4TDP1THRBSMN1; SMN2
SCHEMBL4410768 0.78 TDP1 (0.50) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL7872556 0.76 ALDH1A1 (0.48) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL8427287 0.76 TAAR1 (0.59) ALDH1A1TDP1KDM4ETAAR1NPC1
SCHEMBL14730130 0.76 TDP1 (0.48) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL4001757 0.74 ALOX15 (0.56) ALDH1A1CYP3A4TDP1ALOX15TP53
SCHEMBL29617187 0.74 ALOX15 (0.56) ALDH1A1CYP3A4TDP1ALOX15TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1053239-B1 GLUCOCORTICOID-SELECTIVE ANTI-INFLAMMATORY AGENTS ABBOTT LAB (US) 2003-01-08 EP claimed
EP-3344339-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO Dow AgroSciences LLC (US) 2018-07-11 EP disclosed
EP-3344599-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO Dow Agrosciences LLC (US) 2018-07-11 EP disclosed
EP-3344600-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO Dow Agrosciences LLC (US) 2018-07-11 EP disclosed
WO-2017040191-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2017-03-09 WO disclosed
WO-2017040742-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2017-03-09 WO disclosed
WO-2017040194-A1 MOLECULES HAVING PESTICIDAL UTILITY, AND INTERMEDIATES, COMPOSITIONS, AND PROCESSES, RELATED THERETO DOW AGROSCIENCES LLC (US) 2017-03-09 WO disclosed