SCHEMBL6996478

SCHEMBL6996478

CCCCNC(=O)C=C1CCCc2sc(C(=N)N)cc21

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.33
CYP1A2 P05177 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP2C9 P11712 1/20 0.33
KDM4E B2RXH2 2/20 0.33
HPGD P15428 2/20 0.33
POLB P06746 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
RAB9A P51151 2/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
MAPK10 P53779 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
CYP3A4 P08684 1/20 0.30
GAA P10253 1/20 0.30
ALOX15 P16050 2/20 0.30
CSNK2A2 P19784 1/20 0.30
KDR P35968 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6996475 1.00 ALDH1A1 (0.33) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6990213 0.88 DAO (0.41) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6990211 0.88 DAO (0.41) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6991835 0.86 ALDH1A1 (0.36) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6991832 0.86 ALDH1A1 (0.36) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6997601 0.76 HTT (0.44) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
SCHEMBL6997598 0.76 HTT (0.44) ALDH1A1CYP1A2CYP2C19CYP2C9KDM4E
Hydrochloric Acid SCHEMBL7972762 0.75 C1S (0.33) POLBTDP1
Hydrochloric Acid SCHEMBL7972765 0.75 C1S (0.33) POLBTDP1
Trifluoroacetic Acid SCHEMBL6993161 0.70 C1S (0.31) ALDH1A1CYP1A2CYP2C19HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0927177-B1 NOVEL BENZOTHIOPHENE DERIVATIVES, THEIR PREPARATION AND USE AS UROKINASE INHIBITORS FUJISAWA PHARMACEUTICAL CO (JP) 2003-11-26 EP disclosed
US-6274619-B1 FUSED AMIDINO TYPE COMPOUNDS SUCH AS 4-(N-BUTYLCARBAMOYLMETHYLIDENE)-2-AMIDINO-4,5,6,7-TETRAHYDROBE NZO(B)THIOPHENE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2001-08-14 US disclosed
US-6093710-A AN ENZYME INHIBITOR TREATING ANGIOGENESIS, ARTHRITIS, INFLAMMATION, METASTASIS, OSTEOPOROSIS, TUMORSANGIOGENESIS-DEPENDENT RETINOPATHIES, CONTRACEPTIVE FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-07-25 US disclosed